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(1S,5R)-3-(5-acetyl-4-methylpyrimidin-2-yl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-methoxyphenyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1H-pyrazole-4-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(3-methoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-hydroxy-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)acetamide
(3R,4R)-3-cyclopropyl-4-methyl-1-(2-methyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-ol
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
1-[4-(1H-pyrazol-1-yl)phenyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-[(2-fluorophenyl)methyl]-N-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-N-methylpiperidin-3-amine
3-methoxy-1-[2-oxo-2-(2-phenylpyrrolidin-1-yl)ethyl]-1,2-dihydropyridin-2-one
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(4-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{1-[1-(3,4-difluorophenyl)piperidin-4-yl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
4-[4-(2-methoxyethoxy)phenyl]-6-methylpyrimidin-2-amine
1-[(2-chloro-6-fluorophenyl)methyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
3-amino-3-(3,4-dimethoxyphenyl)-N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
5-fluoro-6-methyl-2-(4-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-cyclopropyl-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}cyclohexanecarboxamide
1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
N-(1H-1,3-benzodiazol-2-yl)-2-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]acetamide
1-{[1-(ethoxymethyl)cyclobutyl]methyl}-5-oxopyrrolidine-3-carboxylic acid
N,2,5-trimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}furan-3-carboxamide
2-benzyl-9-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(1S,5S)-3-{[4-(cyclopentyloxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-[2-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-(4-methylphenoxy)piperidine
methyl (2S,4S,5R)-4-(cyclopentylcarbamoyl)-5-(2-fluorophenyl)-1-methylpyrrolidine-2-carboxylate
5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-(thiolan-3-yl)pyridin-2-amine
4-(2-fluorophenoxy)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
methyl 1-benzyl-5-({[4-(2-hydroxyethoxy)phenyl]methyl}amino)-3-(oxolane-2-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(4-{[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-4,6-dimethylpyridine-3-carbonitrile
(4aS,7aR)-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-4-pentyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,4-dimethoxy-5-(1H-pyrazol-3-yl)pyrimidine
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-3-(furan-2-yl)propanamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-(morpholin-4-yl)butanamide
1-(4-methoxyphenyl)-4-{1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}piperazine
N-(2H-1,3-benzodioxol-5-yl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
N3-[(3-fluorophenyl)methyl]-N5-methyl-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-methyl-N-[2-(4-methylphenoxy)ethyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
2-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-cyclopropyl-3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}propanamide
ethyl 4-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]piperazine-1-carboxylate
(1R,5R)-N,N-dimethyl-6-[4-(4-methylphenyl)-4-oxobutyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
7-cyclopentyl-2-(5,6-dimethylpyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 1-{3-[4-(4-ethylpiperazin-1-yl)piperidine-1-carbonyl]-6-(thiophen-2-yl)pyridin-2-yl}piperidine-3-carboxylate
3-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenol
2-(carbamoylamino)-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}acetamide
1-methanesulfonyl-N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}piperidin-4-amine
N-(2-{1-[(8-chloroquinolin-2-yl)methyl]piperidin-3-yl}ethyl)acetamide
4-[2-(4-fluorophenoxy)ethyl]-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-5-one
3-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-9-methoxy-N-(3-methylbutyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]cyclohex-3-ene-1-carboxamide