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(2S,4R)-N,N-diethyl-1-methyl-4-[3-(1-methyl-1H-pyrazol-4-yl)propanamido]pyrrolidine-2-carboxamide
[3-(hydroxymethyl)-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl]methanol
1-(4-chloro-2-fluorobenzoyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine
6-(1H-1,3-benzodiazol-1-yl)-3,4-dihydroquinazolin-4-one
4-{2-[2-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-5-oxopyrrolidin-1-yl]ethyl}benzene-1-sulfonamide
(4S)-3-[(3,4-dichlorophenyl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
8-[3-(ethylsulfanyl)propanoyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(2S)-1-hydroxybutan-2-yl]-1,3-oxazole-4-carboxamide
(3R,4S)-4-(5-methylfuran-2-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-amine
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{5-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
3-ethyl-3-(4-hydroxybutyl)-1-(3-methoxy-4-methylphenyl)urea
5-{[(4-fluorophenyl)methyl](pyridin-2-ylmethyl)carbamoyl}thiophene-2-carboxylic acid
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(3-hydroxypiperidin-1-yl)-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
N-{[5-(2,3-dihydroxypropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-ethyl-N-(2-hydroxyethyl)piperidine-3-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-methoxy-N,4-dimethylquinazolin-2-amine
1-[4-(pyrazin-2-yl)piperazin-1-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
4-(5-methyl-4-phenyl-1H-imidazol-2-yl)-1-[(4-methylphenyl)methyl]pyrrolidin-2-one
(2S,4S)-4-amino-1-[2-(2,4-dioxoimidazolidin-1-yl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-oxazole-4-carboxamide
3-(3-hydroxyquinoxalin-2-yl)-1-[2-(pyridin-3-yl)pyrrolidin-1-yl]propan-1-one
N4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-6-methylpyrimidine-2,4-diamine
6-{[1-(thiomorpholin-4-yl)hex-5-en-2-yl]oxy}pyridine-3-carbonitrile
6-(benzyloxy)-1-cyclohexyl-4-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-1,4-diazepan-2-one
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[(3-chlorophenyl)methyl]acetamide
[(1,2-dimethyl-1H-imidazol-5-yl)methyl](methyl)[(1-phenyl-1H-pyrazol-4-yl)methyl]amine
N-(2-chlorophenyl)-3-[1-(oxan-4-yl)piperidin-4-yl]propanamide
1-(2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetyl)-N,N-diethylpiperidine-4-carboxamide
2-cyclopropyl-N-[(2-methylphenyl)methyl]-6-oxo-N-(oxolan-2-ylmethyl)-1,6-dihydropyrimidine-5-carboxamide
2-(2,3-dihydro-1H-inden-2-yl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
[2-(1H-imidazol-4-yl)ethyl]({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
2-(2-hydroxyphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
N-(prop-2-en-1-yl)-4-[(pyridin-2-ylsulfanyl)methyl]-N-(pyridin-3-ylmethyl)benzamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
methyl 2-[(cyclopropylmethyl)(propyl)sulfamoyl]-6-(1,2,5-thiadiazole-3-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(5-chlorofuran-2-carbonyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-(1,3-dioxolan-2-ylmethyl)-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2,2-dimethyl-6-[3-(5-methyl-2-{[2-(morpholin-4-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidine-1-carbonyl]-3,4-dihydro-2H-pyran-4-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[3-(1H-imidazol-1-yl)propyl]-5-methoxybenzamide
3-amino-N-({1-[(3,5-difluorophenyl)methyl]pyrrolidin-3-yl}methyl)benzamide
4-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]morpholine
N-[(5-fluoro-1H-indol-2-yl)methyl]-N,5-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
[1-(2,5-dimethylpyrimidin-4-yl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
4-[(1S,2R)-2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-1-hydroxypropyl]phenol
4-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}morpholine
3-(1-benzyl-1H-imidazol-2-yl)-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
1-(4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)ethan-1-one