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1-[1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-1,2,3,6-tetrahydropyridin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
2,4-dimethoxy-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
(2S)-2-acetamido-3-(1H-imidazol-4-yl)-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]propanamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[(2,2,6,6-tetramethylpiperidin-4-yl)amino]methyl}piperidin-2-one
2-(oxolan-2-ylmethoxy)-1-{4-[(prop-2-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
2-[(5-methylpyrazin-2-yl)methyl]-9-(propane-1-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]piperidin-1-yl}pyrazine
1-(2-ethoxyethyl)-N,N-diethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-{[2-(difluoromethoxy)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,1,3-trimethyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(azepan-1-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
[4-benzyl-1-(naphthalen-1-ylmethyl)piperidin-4-yl]methanol
6-chloro-N-cyclopropyl-3-fluoro-N-[(3-hydroxyphenyl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl](quinoxalin-2-ylmethyl)amine
8-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 2-{4-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]-2-methoxyphenoxy}acetate
2-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)-N-propyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
dimethyl(3-{2-[1-(3-methylpyridin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
6-[2-(4,5,6,7-tetrahydro-1H-indazol-3-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazole-5-carbonyl]-2-methyl-2,3-dihydro-1H-indole
2-amino-N-[(3R,4S)-4-cyclopropyl-1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]pyrrolidin-3-yl]acetamide
[5-fluoro-7-(6-methoxypyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-({2-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)azepan-4-ol
1-benzoyl-4-[4-(methylamino)pyrimidin-2-yl]-1,4-diazepan-6-ol
4-[(2R,5R)-2,5-dimethylpyrrolidine-1-carbonyl]-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole
[(3-chloro-5-fluorophenyl)methyl](methyl)[4-(morpholin-4-yl)butyl]amine
2-[(4-fluorophenyl)methyl]-N-[4-(methylsulfanyl)phenyl]morpholine-4-carboxamide
1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]azocane
N-methyl-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-(pyridin-2-ylmethyl)propanamide
N-[2-(3-ethoxyphenoxy)ethyl]-N-methyl-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
2-(5-chloro-2-methoxypyridin-4-yl)-3-(pyrrolidin-1-yl)pyrazine
2-(2-methyl-1H-imidazol-1-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
N-[(3-methylphenyl)methyl]-N-(propan-2-yl)-3-(1H-1,2,4-triazol-1-yl)propanamide
(1R,5R)-6-methyl-3-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
3-[(3R,4S)-1-(2,5-dimethylfuran-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazine
3-{[(3S,4S)-3-hydroxy-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-1-yl]methyl}-4H-chromen-4-one
6-methoxy-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-methyl-4-{[8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}-1H-pyrrole-2-carbonitrile
7-chloro-3-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3,4-dihydroquinazolin-4-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
5-[4-(azepane-1-carbonyl)-5,7-dimethylquinolin-2-yl]-N-methylpyrimidin-2-amine
2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-6-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1H-indole
4-(1H-1,3-benzodiazol-1-yl)-1-(1,3-thiazole-4-carbonyl)piperidine-4-carboxylic acid
(3aS,6aS)-5-(1,4-dithiepan-6-yl)-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-chloro-4-methoxyphenyl)-3-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]propanamide
2-[3-(3-fluorophenyl)-1,2-oxazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide