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methyl 3-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2S)-4-methyl-2-({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amino)pentanamide
2-[2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-1,3-benzoxazole
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
3-methyl-7-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
6-[1-(5-methoxy-1-methyl-1H-indole-2-carbonyl)piperidin-3-yl]pyrimidin-4-ol
(4aS,8aR)-6-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
8-fluoro-2-[4-(4-methylphenyl)-3-oxopiperazine-1-carbonyl]-1,4-dihydroquinolin-4-one
N-methyl-N-propyl-2-{4-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]morpholin-3-yl}acetamide
1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-3-(3-methoxyphenoxy)azetidine
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(4-chlorophenoxy)pyridine-3-carboxamide
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-2,6-dimethylpyridine-4-carboxamide
2-(4-ethoxyphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
4-(2-methoxy-4-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(2,3-dihydro-1H-inden-1-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]acetamide
5-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
1-(4-{[2-(1H-pyrazol-4-yl)ethyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(3S,9aR)-3-(cyclohexylmethyl)-8-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
N-cyclopropyl-2-(2,5-dimethoxyphenyl)-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}acetamide
N-[2-(azepan-1-yl)ethyl]-N-methyl-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-[2-(2,5-dimethoxyphenyl)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
7-(2-amino-1,3-benzothiazole-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(3-methoxypropyl)-8-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-phenylpiperidine-1-carboxamide
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-{2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-N-(1-phenylethyl)acetamide
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-(2-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)-2-methoxyethan-1-one
5-{1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1H-imidazol-2-yl}-N,N-dimethylpyrimidin-2-amine
(8R,9aS)-8-hydroxy-2-[3-(1H-indazol-1-yl)propyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
(3R,4R)-3-cyclobutyl-1-(3-methoxybenzenesulfonyl)-4-methylpyrrolidin-3-ol
4-hydroxy-2-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
2-[4-(1H-indol-2-ylmethyl)-1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
2-(4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
4-[(2H-1,3-benzodioxol-4-ylmethyl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}furan-2-carboxamide
3-methyl-5-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-2,3-dihydro-1,3-benzoxazol-2-one
2-(4-{[3-(3-chlorophenyl)phenyl]carbamoyl}piperidin-1-yl)acetic acid
3-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
1-[(2-chlorophenyl)methyl]-4-{[(4-fluoro-3-methoxyphenyl)methyl]amino}pyrrolidin-2-one
N-cyclopentyl-3-[(2-fluorophenyl)formamido]-N-(prop-2-en-1-yl)propanamide
(3S,4R)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2-(4-fluoro-3-methylphenyl)-2-(4-hydroxypiperidin-1-yl)acetic acid
2-(2-fluorophenyl)-8-methoxy-5-[(4-methyl-1H-imidazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
5-(dimethylamino)-2-[(2-methoxypyridin-3-yl)methyl]-2,3-dihydropyridazin-3-one
N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-4-methylpyrimidin-2-amine
N-cyclohexyl-3-({[2-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]carbamoyl}amino)propanamide
N-{1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]piperidin-4-yl}methanesulfonamide