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3-(3,4-dimethylphenyl)-N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)propanamide
4-({[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl](methyl)amino}methyl)-1-methylpyrrolidin-2-one
2-(4-methanesulfonylphenyl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
5-[benzyl(methyl)amino]-2-(3-hydroxypropyl)-2,3-dihydropyridazin-3-one
4-hydroxy-1-[3-(piperidine-1-carbonyl)pyridin-2-yl]piperidine-4-carboxylic acid
6-(1,4-diazepan-1-yl)-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]pyridine-3-carboxamide
5-{[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]methyl}-2-methoxyphenol
8-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[1-(2,5-difluorophenyl)cyclopropyl]-6-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
(2S,4R)-1-[(3-ethoxy-4-methoxyphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
(3S,7S)-5-(5-ethyl-1H-pyrrole-2-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-1-methylpiperidine
4-(3-{[(4-phenylphenyl)formamido]methyl}piperidine-1-carbonyl)pyridin-1-ium-1-olate
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-(methylsulfanyl)propanamide
1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-N-(2-phenylethyl)piperidin-3-amine
1-(thiophen-3-ylmethyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{2-[4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
6-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N,N-dimethylpyridine-3-carboxamide
2-[1-(6-aminopyridin-3-yl)-4-methyl-1H-1,3-benzodiazol-2-yl]ethan-1-ol
1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-N,N-dimethylpiperidin-3-amine
1-ethyl-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
methyl 4-{[5-(1H-1,3-benzodiazol-1-ylmethyl)-1,2-oxazol-3-yl]formamido}butanoate
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-3-(piperidin-3-yl)benzamide
N-methyl-3-(2-methyl-1H-imidazol-1-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
N-[1-(methylcarbamoyl)cyclohexyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N,5-dimethyl-2-phenyl-1H-imidazole-4-carboxamide
(2S,4R)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
1'-[(5-acetylthiophen-3-yl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
5-(2H-1,3-benzodioxol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
3-({methyl[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}methyl)pyridin-2-amine
2-(2-{[1-(1-methyl-1H-pyrazol-4-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-(5-ethyl-1,3,4-thiadiazol-2-yl)-1-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]urea
2-[3-(2,4-difluorophenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
N-[1-({2-oxo-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-3-yl}methyl)piperidin-4-yl]methanesulfonamide
2-[3-oxo-9-(3-phenylbutyl)-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
3-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
1-(3-chloro-4-methoxyphenyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
4-oxo-N-(oxolan-2-ylmethyl)-N-propyl-3,4-dihydroquinazoline-2-carboxamide
2-(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)propan-2-ol
2-{1-[(4-methylphenyl)methyl]-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
4-(5-methylpyridin-2-yl)-1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-ol
[3-(3,4,5-trimethoxyphenyl)phenyl]methanol
3-[(3R,4S)-1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]-4-phenoxypiperidine-4-carboxylic acid
(4aR,7aS)-1-ethyl-4-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[5-(3,4-difluorophenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
4-hydroxy-N-{[4-(2-methoxyethoxy)phenyl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide