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diethyl({2-[4-(1-ethyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]ethyl})amine
(1S,4S)-2-benzyl-5-(3-propyl-1H-pyrazole-5-carbonyl)-2,5-diazabicyclo[2.2.1]heptane
1-(4-{[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]amino}piperidin-1-yl)butan-1-one
N-(2,4-dimethoxyphenyl)-3-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}propanamide
5-(2,6-dimethoxyphenyl)-3-[4-(4-methoxyphenoxy)piperidin-1-yl]-1,2,4-triazine
2-[2-(3-hydroxypiperidin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
3-[(3R,4S)-1-(1H-imidazol-2-ylmethyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(4-fluorophenyl)-1,4-diazepane
9-{[4-(methylsulfanyl)phenyl]methyl}-3-oxa-9-azaspiro[5.5]undecane
{5-[({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]furan-2-yl}methanol
[4-benzyl-1-(5-fluoro-2-methylbenzenesulfonyl)piperidin-4-yl]methanol
3-[1-(5-chlorothiophene-2-carbonyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-1-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethan-1-one
4-{1-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperidin-4-yl}thiomorpholine
4-({5-chloro-2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)thiomorpholine
1-(pyridin-3-ylmethyl)-4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-1,4-diazepane
(4aR,8aR)-2-[(2-chlorophenyl)methyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
8-(1,3-benzothiazol-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[2-(1H-indol-3-yl)ethyl]-N-(pyridin-3-ylmethyl)oxane-2-carboxamide
1-[(2-ethylpyrimidin-5-yl)methyl]-4-(2-fluoro-5-methylphenoxy)piperidine-4-carboxylic acid
N-[(8-methoxyquinolin-5-yl)methyl]-N,6-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl][(2-fluorophenyl)methyl]methylamine
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-(1-aminocyclobutanecarbonyl)-4-(2-fluoro-5-methylphenoxy)piperidine-4-carboxylic acid
methyl 2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetate
1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
5-hydroxy-6-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidine-1-carbonyl]-2-(4-methylphenyl)-2,3-dihydropyridazin-3-one
2-{1-benzyl-4-[(8-methoxy-2H-chromen-3-yl)methyl]piperazin-2-yl}ethan-1-ol
1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid
(3R,4R)-4-cyclopropyl-1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-3-methylpiperidin-4-ol
(1S,5R)-3-methyl-6-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
ethyl 2-(1-{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-2-yl)acetate
N-methyl-N-[2-(oxan-2-yl)ethyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-[2-(thiophen-2-yl)ethyl]propanamide
4-chloro-2-{[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]methyl}phenol
2-[(1-ethylpyrrolidin-2-yl)methyl]-1,2-dihydroisoquinolin-1-one
3-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-1-(2-fluoro-4-methoxyphenyl)urea
2-[3-cyclopentyl-5-(3-phenylpropyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
methyl 2-(4-{[3-(methylcarbamoyl)-1,2,4-oxadiazol-5-yl]methyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl)acetate
2-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]benzene-1,3-diol
2-cyclopropyl-8-[(3-ethoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-[4-(5-methylthiophen-2-yl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
1-[(2-fluorophenyl)methyl]-3-{2-[(3S)-3-hydroxypyrrolidin-1-yl]-2-oxoethyl}-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-[3-(3-ethylphenoxy)propyl]-N-methyl-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
1-[cyclohexyl(methyl)amino]-3-[2-({methyl[3-(pyrrolidin-1-yl)propyl]amino}methyl)phenoxy]propan-2-ol
2-{4-[(4-fluorophenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{[5-(2,3-dihydro-1H-inden-1-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-methylpiperazine
9-(2-methyl-1,3-thiazole-4-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}-N-[2-(pyrazin-2-yl)ethyl]benzamide