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3-(3-chloro-1,2-oxazol-5-yl)-1-[3-(2-methylphenoxy)azetidin-1-yl]propan-1-one
3-(4-chloro-1H-pyrazol-1-yl)-1-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]propan-1-one
(1R,7S)-3-(2-ethoxyethyl)-6-(3-oxopiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetic acid
4,6-dimethyl-3-{[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-indol-2-one
8-methoxy-N-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
2-[4-(2-chlorophenoxy)piperidine-1-carbonyl]-N,N-dimethylaniline
4-{5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-imidazol-2-yl]thiophen-2-yl}-2-methylbut-3-yn-2-ol
1-(4-fluoro-3-methoxyphenyl)-2-{[5-(methoxymethyl)furan-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
(1R,5S,6S)-6-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-3-azabicyclo[3.1.0]hexane
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
(3S,4R)-1-[2-(4-fluorophenyl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
2-(2H-1,3-benzodioxol-5-yl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
3-(3-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}-1H-indol-1-yl)propanamide
2-(cyclopropylmethyl)-7-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(thiophen-3-yl)propan-2-yl]benzamide
N-({3-[(3-chlorophenyl)methyl]-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl}methyl)acetamide
(4aS,8aR)-6-(2-ethoxypyridine-3-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
(1S,2S,3R,4R)-3-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]bicyclo[2.2.1]heptan-2-amine
{2-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-oxoethyl}urea
1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(4-fluorophenyl)sulfanyl]piperidine
2-(1-methyl-1H-pyrazol-4-yl)-4-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]quinoline
5-{[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2,7-dioxo-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1,3-diazepane-4-carboxamide
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-1,3-thiazole-4-carboxamide
(4aS,8aR)-6-[4-(2-aminoethyl)benzoyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-cyclopropyl-3-(5-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanamide
4-{[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]methyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N-[5-(furan-2-yl)-1,3,4-thiadiazol-2-yl]-4-methyl-1,4-diazepane-1-carboxamide
2-chloro-N-[2-(2-methyl-1H-pyrrole-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
2-cyclohexyl-6-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
(3aR,6aR)-2-methyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
2-benzyl-9-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazine-1-carbonyl}cyclopropane-1-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
2-methyl-5-[2-(oxan-2-ylmethyl)phenyl]-1,3,4-thiadiazole
N-[(4-cyanophenyl)methyl]-3-{[(4-fluorophenyl)methyl]sulfanyl}propanamide
2-(dimethylamino)-1-[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]ethan-1-one
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)propanamide
N-(2-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-2-yl}ethyl)acetamide
3-(2-methylpyrimidin-4-yl)-4H-chromen-4-one
6-methyl-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]pyridazin-3-amine
4-[1-(1-cyclopropylethyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-methyl-3-phenyl-1H-pyrazole
2-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
(2S)-1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxamide
(2E)-N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(3-fluorophenyl)prop-2-enamide
2-(2-hydroxyethyl)-9-[(4-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(3-chlorobenzoyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol