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(4aS,7aR)-1-(1H-imidazol-4-ylmethyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 1-{1-[4-(3-phenylpropanamido)phenyl]piperidin-4-yl}piperidine-4-carboxylate
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-3-(1H-pyrazol-1-yl)propanamide
2-(4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
6-methyl-5-{5-[4-(propan-2-yl)-1,3-thiazol-2-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
7-[2-(3,4-dimethoxyphenyl)acetyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-phenyl-3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carboxamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one
2-(1-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-imidazol-2-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole
(4aS,8aR)-6-[2-(5-amino-1,3,4-thiadiazol-2-yl)acetyl]-1-butyl-decahydro-1,6-naphthyridin-2-one
2-(adamantan-1-yl)-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
3-[3-(1-methylpiperidin-4-yl)-4H-1,2,4-triazol-4-yl]pyridine
4-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-{1-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
2-(2-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}ethoxy)ethan-1-ol
1-(2,3-dihydro-1H-inden-2-yl)-4-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-1,4-diazepane
2-(3-phenylpropyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,3-benzoxazole-5-carboxamide
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(4-fluorophenyl)methyl]piperidine
2-(1,2-benzoxazol-3-yl)-1-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]ethan-1-one
2-(2-chlorophenyl)-5-methyl-4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1,3-oxazole
1-(1-cyclohexylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-benzyl-N,1-dimethyl-5-{[(6-methylpyridin-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(4-aminoazepane-1-carbonyl)-4-fluorobenzene-1-sulfonamide
3-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-pyrazol-5-amine
N-[2-(2-chlorophenyl)-1-[1-(2-methylpropyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
2-amino-4-(1-methyl-1H-pyrazol-4-yl)-5H,6H,7H-pyrrolo[2,3-h]quinoline-3-carbonitrile
5-ethyl-4-({3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}methyl)furan-2-carboxamide
N-benzyl-N-methyl-3-{[(3-phenylpropyl)amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
2-(dimethylamino)-N,4-dimethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}pyrimidine-5-carboxamide
3-cyclopropyl-5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]-1H-1,2,4-triazole
N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}-9-methyl-9H-carbazole-3-carboxamide
1-methyl-8-[(1-methyl-1H-indol-2-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(4aS,8aR)-6-(1H-imidazol-2-ylmethyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
1-[(4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)methyl]-1H-1,2,3,4-tetrazole
1-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazole
N-(3-cyanothiophen-2-yl)-3-{[2-(methoxymethyl)piperidin-1-yl]methyl}benzamide
2-[1-(propan-2-yl)piperidin-4-yl]-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethan-1-one
1-(4-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
2-[5-(4-methanesulfonylphenyl)-3-methyl-1H-1,2,4-triazol-1-yl]acetic acid
2-[(4-chlorophenyl)methyl]-5-{7-ethyl-2,7-diazaspiro[4.4]nonane-2-carbonyl}-1,3-benzoxazole
(1R,5S)-6-[5-(4-chloro-2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-6-azabicyclo[3.2.1]octane
2,2-dimethyl-1-(1-methyl-4-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,4,9-triazaspiro[5.5]undecan-9-yl)propan-1-one
N-[4-(furan-2-yl)phenyl]-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidine-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(morpholin-4-yl)benzamide
1-{4-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}imidazolidine-2,4-dione
1-{4-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]thiophen-2-yl}ethan-1-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
(3aR,6aR)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(2-methoxyacetyl)-N-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1-(propan-2-yl)piperidine-4-carboxamide