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1-{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
1-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)ethan-1-one
2-[5-(3-fluoro-4-methoxyphenyl)-1H-indol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
dimethyl(2-{2-[1-(3-methylpyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-2H-1,3-benzodioxole-5-carboxamide
N-(2-hydroxyethyl)-1-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxamide
4-[(2-fluorophenyl)methyl]-3-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-2-one
5-amino-3-(6-fluoro-1-methyl-1H-indol-3-yl)-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
ethyl 3-[2-(pyridin-3-yl)pyrimidine-5-amido]azepane-1-carboxylate
1-[1-(2-ethylbutanoyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[3-(pyrrolidin-1-yl)propyl]benzamide
(2R,3R)-3-[methyl(propyl)amino]-1'-(4-methylpyridin-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
3-{2-[(3-methoxyphenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanoic acid
2-hydroxy-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-(3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-oxopropyl)azepan-2-one
4-{[(2-methoxyphenyl)methyl]amino}-5-methyl-N,N-bis(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-4-oxo-N-(pyridin-4-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-3-cyano-5-fluorobenzamide
N-({1-[(2-methoxypyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)-3-methylfuran-2-carboxamide
2-methyl-9-{[4-(2-methylpropyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-{3-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]phenyl}imidazolidin-2-one
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(1-methylcyclopropanecarbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[3-(1H-imidazol-1-yl)propyl]-4-(1H-pyrazol-3-yl)benzamide
9-(2-amino-2-methylpropanoyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
7-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1-[1-(1-aminocyclopropanecarbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-5-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
N-[(2R,4R,6S)-2-(propan-2-yl)-6-[3-(1H-pyrazol-1-ylmethyl)phenyl]oxan-4-yl]acetamide
N,1-dimethyl-N-{1-[1-(2-oxo-2H-chromene-3-carbonyl)piperidin-4-yl]-2-phenylethyl}-1H-pyrazole-3-carboxamide
N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
[2-(tert-butylsulfanyl)ethyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
ethyl 4-{4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}piperidine-1-carboxylate
2-methyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
5-[2-(quinolin-4-yl)-1H-imidazol-1-yl]pyridine-3-carboxylic acid
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-4-(1H-imidazol-1-yl)butan-1-one
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]but-2-ynamide
4-ethyl-1-[(2-fluorophenyl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,7,8-trimethylquinoline-4-carboxamide
N-[(4-fluorophenyl)methyl]-3-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]propanamide
5-fluoro-2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-3-methyl-1H-indole
3-{1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
(5S,9aS,9bS)-5-(1-methyl-3-phenyl-1H-pyrazol-4-yl)-2-(1-methylpiperidin-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(5-methylfuran-2-yl)methyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)quinazolin-4-amine
5-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}pyrimidine-2,4-diol
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]morpholine-4-sulfonamide
N-{2-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]ethyl}acetamide
N-ethyl-2-(7-methyl-2-oxo-2H-chromen-4-yl)-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
N-{[7-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1-phenylmethanesulfonamide