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1-[(1-{[1-(pyrimidin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]-1,4-diazepane
{5-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]furan-2-yl}methanol
[(3-{1-butyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]dimethylamine
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-3-(pyrazin-2-yl)propanamide
3-(furan-2-yl)-3-phenyl-N-(pyridin-3-ylmethyl)propanamide
3-methoxy-N-{2-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}propanamide
3-{2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamido}-N-phenylpropanamide
5-ethyl-N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
1-[(4aR,8aR)-4a-hydroxy-7-methanesulfonyl-decahydro-2,7-naphthyridin-2-yl]-2-(2H-1,3-benzodioxol-5-yl)ethan-1-one
2-methyl-N-[(1s,4s)-4-aminocyclohexyl]-1-benzofuran-7-carboxamide
(1H-imidazol-4-ylmethyl)(methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
4-(1H-pyrazol-4-yl)-N-[2-(pyridin-2-yl)ethyl]butanamide
3-ethyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}urea
2-({[(6-chloropyridin-3-yl)methyl](methyl)amino}methyl)pyridine-3-carboxylic acid
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
(3S,4S)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
1-ethyl-4-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-1,2-dihydropyridin-2-one
N-[(2R,4R,6S)-2-(3,5-difluorophenyl)-6-(2,5-dimethoxyphenyl)oxan-4-yl]acetamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(1,2-oxazole-3-carbonyl)piperidine
3-(3-chloro-1,2-oxazol-5-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
1-ethyl-5-[(1H-1,2,4-triazol-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-(oxan-4-yl)-2-{4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]morpholin-3-yl}acetamide
1-[2-methyl-4-({2-[1-(2-methylpropyl)piperidin-2-yl]ethyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
(4aR,7aS)-1-[2-(2,3-dihydro-1H-isoindol-2-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2,2-dimethylpropyl)-3-hydroxy-3-(piperidin-1-ylmethyl)piperidin-2-one
7-methyl-2-(1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(2,3,4-trimethoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
5-(azepane-1-carbonyl)-N-ethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
1-[benzyl(methyl)amino]-3-{4-[(4-fluoropiperidin-1-yl)methyl]phenoxy}propan-2-ol
(2S,4S)-4-amino-1-(2,1,3-benzoxadiazole-5-carbonyl)pyrrolidine-2-carboxylic acid
5-butyl-1-(2-methoxyphenyl)-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperazin-2-one
methyl(2-phenoxyethyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
4-benzyl-1-(ethanesulfonyl)-3-ethyl-1,4-diazepan-5-one
1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(4H-1,2,4-triazol-4-yl)propan-1-one
N,N,4-trimethyl-5-[3-(pyridin-3-yl)azetidine-1-carbonyl]pyrimidin-2-amine
3-[(3R,4S)-1-(dimethyl-1,2-oxazole-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(1S,5R)-6-[(4-methoxynaphthalen-1-yl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-(3-hydroxypyrrolidin-1-yl)-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1-ethyl-5-oxopyrrolidine-3-carboxamide
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
3-(2-ethoxyethyl)-2-oxo-1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(3-methyl-1H-pyrazol-1-yl)propanamide
6-[1-(carbamoylmethyl)piperidine-3-carbonyl]-N,1-dimethyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
4-methoxy-6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyrimidine
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(3-methylbutyl)-1,2-oxazole-3-carboxamide