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3-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]phenol
3-(1,2-oxazinan-2-yl)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]propanamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[(4,6-dimethylpyrimidin-2-yl)methyl]amine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(2,5-dioxoimidazolidin-1-yl)acetamide
3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-8-(piperidin-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-cyclopentyl-4-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-4-sulfamoylbenzamide
1-methyl-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1H-pyrazole-5-carboxamide
1-ethyl-8-{[4-(methylsulfanyl)phenyl]methyl}-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(3-chloro-4-hydroxyphenyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)acetamide
1-(2-methoxyethyl)-3-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1-(1,3-thiazol-2-ylmethyl)urea
4-(5-chloro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(adamantan-2-yl)-4-[(2S,4S)-1-[(2-chloro-6-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]piperazine
(1S,3R)-3-amino-N-(4-chloro-3-fluorophenyl)cyclopentane-1-carboxamide
N-(2-hydroxy-2-phenylethyl)-2,4-dimethyl-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
N-cyclopropyl-5-(2-fluorophenoxymethyl)-N-(oxan-4-yl)-1H-pyrazole-3-carboxamide
4-benzyl-3-ethyl-1-(thiophen-2-ylmethyl)-1,4-diazepan-5-one
N-({5-[(4-fluoro-2-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[1-(4-fluorophenyl)ethyl]propanamide
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
1-(2-methoxyethyl)-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
4-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
{[4-(butan-2-yloxy)-3-ethoxyphenyl]methyl}[(5-methylpyrazin-2-yl)methyl]amine
ethyl 2-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}-1,3-oxazole-4-carboxylate
(3S,4R)-1-(cyclobutylmethyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
4-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
5-{[(1-benzofuran-2-ylmethyl)(propan-2-yl)amino]methyl}pyrrolidin-2-one
2-[2-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy]-1-[4-(2,3-dimethylphenyl)piperazin-1-yl]ethan-1-one
4-(2-chlorophenoxy)-1-(4-methyl-1,3-thiazol-2-yl)piperidine
6-(3-chlorophenyl)-N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
(4aS,7aR)-1-(2-butoxyacetyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-cyano-N-[2-fluoro-3-(trifluoromethyl)phenyl]piperidine-1-carboxamide
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-ethyl-N-methylpropanamide
N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-3-(4-methylphenyl)propanamide
1-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidine-1-carboxamide
(2S,3R)-2-{[(6,7-dimethyl-2-oxo-2H-chromen-4-yl)methyl]amino}-3-hydroxybutanamide
3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-N-(5-methylpyrazin-2-yl)benzamide
2-(4-chlorophenyl)-4-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]morpholine
4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-2-(1-ethyl-1H-pyrazol-4-yl)-6-methylquinoline
2-(3-methoxyphenyl)-6-[4-(pyrrolidin-1-yl)piperidine-1-carbonyl]-1,3-benzoxazole
3-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-2-methoxyquinoline
N-(1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)methanesulfonamide
5-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine-2-carbonitrile
2-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-1-(morpholin-4-yl)ethan-1-one