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1-{5-[4-(3-fluorophenoxy)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
5-{[(2,3-dihydro-1H-inden-1-yl)amino]methyl}-N-(4-methoxyphenyl)-1,3-thiazol-2-amine
5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
1-(cyclohexylmethyl)-N-methyl-5-(4-methylpiperazin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[1-(4-methoxyphenyl)-5-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridin-3-yl]-1H-1,2,4-triazol-3-yl]acetamide
3-hexyl-8-{imidazo[1,2-a]pyridine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)thiomorpholine
2-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}pyridine-3-carboxylic acid
N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}-1H-1,2,4-triazole-5-carboxamide
1-(cyclohexylcarbamoyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
5-{10,10-dichlorotricyclo[7.1.0.04,6]decan-5-yl}-3-(2-methylpropyl)-1,2,4-oxadiazole
3-({[(dimethylcarbamoyl)methyl](methyl)amino}methyl)-N-(quinoxalin-6-yl)benzamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
methyl 2-{3-[3-(3-methylpyridin-2-yl)phenyl]-1H-pyrazol-1-yl}propanoate
2-[1-({1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]pyridine
2-(2,5-dioxoimidazolidin-4-yl)-N-[2-(5-methylfuran-2-yl)ethyl]acetamide
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-(1H-indol-3-yl)propan-1-one
N-{[1-(methoxymethyl)cyclopropyl]methyl}-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-2-(trifluoromethyl)benzene-1-sulfonamide
1-[1-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
2-(3-chlorophenyl)-N-(4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}phenyl)acetamide
3-methyl-N-{[1-(3,3,3-trifluoropropyl)pyrrolidin-3-yl]methyl}benzamide
5-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
2-(2H-1,2,3-benzotriazol-2-yl)-N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
1-[6-(3-aminoazepan-1-yl)pyrimidin-4-yl]piperidin-4-ol
3-[1-(3-phenylpropanoyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
3-[5-(quinoxaline-6-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
4-(2-{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}ethyl)morpholine
N-ethyl-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(oxolan-2-ylmethyl)propanamide
N-[2-(dimethylamino)ethyl]-4-{2-methyl-1H-imidazo[4,5-b]pyridin-6-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
3-{2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
3-{2-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N4-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-N6-(propan-2-yl)pyrimidine-4,6-diamine
(3E)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]pent-3-en-1-one
N-(3-fluorophenyl)-3-(1,2,3,6-tetrahydropyridin-1-ylmethyl)benzamide
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-{1,3-dimethyl-4-[3-(piperidin-1-yl)azetidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
3-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aS)-5-(2-chloro-6-fluoro-3-methylbenzoyl)-1-methyl-octahydropyrrolo[3,4-b]pyrrole
1-(propan-2-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
methyl 3-[2-amino-3-cyano-6-(1,3-dimethyl-1H-pyrazol-4-yl)pyridin-4-yl]benzoate
1-({1-[(3-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}methyl)-3-(propan-2-yl)urea
N-{[1-(1H-indole-5-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
4-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1,3-oxazole-5-carboxamide
1-(2-chlorophenyl)-4-{[4-(2-hydroxyethoxy)phenyl]methyl}-5-methylpiperazin-2-one
1'-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2E)-3-(1H-imidazol-4-yl)-1-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]prop-2-en-1-one