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2-tert-butyl-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
N-[(3S,4R)-1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-(4-hydroxyphenyl)-N-{2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
2-butyl-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
4-[(2,5-dichlorophenyl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methylpyrimidin-2-amine
N-[(7-chloro-4-{[(4-fluorophenyl)methyl]amino}quinazolin-2-yl)methyl]propane-2-sulfonamide
1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-4-phenylpiperazine
N-[(2-chlorophenyl)methyl]-5-oxo-N-(prop-2-en-1-yl)hexanamide
4-(morpholin-4-yl)-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]butan-1-one
3-(2-ethylbutyl)-8-(2-methyl-1,3-thiazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[4-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]ethan-1-one
N-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]pyrazin-2-amine
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
1-(4-chlorophenyl)-N-propyl-N-(pyridin-3-ylmethyl)cyclopropane-1-carboxamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
2-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetic acid
N-benzyl-8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-[(3S,4R)-4-amino-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-yl]ethan-1-ol
1-[(4-fluorophenyl)methyl]-4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-2-one
4-(morpholine-3-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)-2,3-dihydro-1H-inden-2-amine
N-cyclopentyl-N'-[2-(pyridin-3-yloxy)propyl]butanediamide
3-[(3R,4S)-1-[(3-chloro-2,6-difluorophenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-4,4,4-trifluorobutan-1-one
{1-[(8-methoxyquinolin-2-yl)methyl]-3-(3-phenylpropyl)piperidin-3-yl}methanol
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[methyl(1,2-oxazol-3-ylmethyl)amino]pyridine-3-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]propan-1-one
1-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-3,3-bis(propan-2-yl)urea
4-(4-methyl-1H-pyrazol-1-yl)-1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidine-4-carboxylic acid
8-acetyl-2-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(hexan-3-yl)-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-(5-methylfuran-2-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
4-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane-2-carbonyl)pyridin-1-ium-1-olate
2-amino-6-ethyl-4-[4-(methylsulfanyl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
5-ethyl-5-[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]imidazolidine-2,4-dione
2-(methoxymethyl)-1-{1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidin-4-yl}-5-(trifluoromethyl)-1H-1,3-benzodiazole
4-(4-ethoxy-3-methylphenyl)-4-oxo-N-(oxolan-2-ylmethyl)butanamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[6-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
(3aR,6aS)-5-{2-[cyclopentyl(methyl)amino]acetyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(1-butyl-1H-imidazol-2-yl)-1-(4-chloro-2-methoxybenzoyl)piperidine
3-(4-hydroxyphenyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
2-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(2-ethoxy-5-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}phenyl)methanol
2,2-dimethyl-1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
2-{3-cyclopentyl-5-[2-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
2-{4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[1-(4-methoxyphenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]cyclobutanecarboxamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-(methylsulfanyl)acetamide
4-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-2-methyl-1H-1,3-benzodiazole