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N-[4-(2-methanesulfonylacetamido)-2-methylphenyl]pentanamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-ol
(2S,4R)-1-[(2,5-dimethylphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
dimethyl[(4-methyl-5-{1-[4-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
5-methyl-4-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-pyrazol-3-one
9-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-1,4,9-triazaspiro[5.5]undecan-5-one
1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4-(3-methylpyridin-2-yl)piperazine
(2S,4S)-4-[(cyclohexylmethyl)amino]-1-(2,3-dihydro-1H-inden-2-yl)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-(1-benzoylpiperidin-4-yl)-3-[(dimethylamino)methyl]pyrrolidin-3-ol
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-{1,3-dioxo-2-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-isoindol-4-yl}-N-(prop-2-en-1-yl)piperidine-3-carboxamide
N-[(3R,4R)-3-hydroxy-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl]pyridine-2-carboxamide
2-{5-[2-(3,4-difluorophenyl)ethyl]-3-ethyl-1H-1,2,4-triazol-1-yl}acetic acid
7-methyl-2-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
N-(5-chloro-2-methoxyphenyl)-3-{1-[(2-ethoxyphenyl)methyl]piperidin-3-yl}propanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,5-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methyl-2,3-dihydro-1-benzofuran-5-carboxamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-2-cyclopropyl-4-hydroxypyrimidine-5-carboxamide
1-methyl-2-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-1H-indole
2-methoxy-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-{5H,6H,7H-cyclopenta[b]pyridin-7-yl}-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-[3-(4-acetylpiperazine-1-carbonyl)piperidin-1-yl]-2-cyclooctyl-2,3-dihydro-1H-isoindole-1,3-dione
1-{[(3R,4R)-4-(hydroxymethyl)-1-(6-methoxy-1-methyl-1H-indole-2-carbonyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
6-ethoxy-3-{[ethyl(oxan-4-yl)amino]methyl}-1,2-dihydroquinolin-2-one
9-(4-hydroxybenzoyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl){[4-(trifluoromethyl)phenyl]methyl}amine
2-[9-(4-cyanopyridin-2-yl)-7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]acetamide
2-[1-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-2-methylbutyl]-2,3-dihydro-1H-isoindol-1-one
2-(4-fluorophenoxymethyl)-4-hydroxy-N-[1-(1H-imidazol-2-yl)ethyl]pyrimidine-5-carboxamide
2-{1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-2-yl}-1,3-benzothiazole
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-4-(1H-pyrrole-2-carbonyl)piperazine
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]acetamide
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1H-indazol-1-yl)ethan-1-one
11-{[(2-fluorophenyl)methyl]amino}-4-[2-(3-methoxyphenyl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[3-hydroxy-3-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(3-methyl-2-oxopentanoyl)piperidin-4-yl]oxy}benzamide
(furan-2-ylmethyl)[(3-methyl-1H-pyrazol-5-yl)methyl](3-methylbutan-2-yl)amine
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
6-{4-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
(5S,9aS,9bS)-5-[3-(benzyloxy)phenyl]-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3aS,6aS)-2-(cyclopropylmethyl)-1-oxo-5-{thieno[3,2-d]pyrimidin-4-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(6-methyl-2-phenylpyrimidin-4-yl)-1,4-diazepan-5-one
1-{[3-(difluoromethoxy)phenyl]methyl}-4-(2,6-dimethylpyridin-4-yl)piperazine
2-(4-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-1,3-benzoxazole
2-(3-methyl-1,2-oxazol-5-yl)-N-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]pyrrolidine-1-carboxamide
1-(4-benzylpiperidin-1-yl)-3-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}propan-1-one
2-(4-methoxyphenyl)-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
3-methyl-8-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one