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(4aR,7aS)-1-{2-[methyl(3-methylbutyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4R)-4-(2,6-difluoro-4-methoxybenzamido)-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]pyrrolidin-3-amine
4-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
1-cyclobutanecarbonyl-N-[1-(6-methylpyridin-3-yl)ethyl]piperidine-4-carboxamide
[(1-ethyl-1H-pyrazol-4-yl)methyl][(2-ethylpyrimidin-4-yl)methyl]methylamine
3-[(3R,4S)-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
1-[(3-chloro-4-methoxyphenyl)methyl]-4-(1-methylpiperidin-4-yl)piperazine
(4aS,8aR)-6-[2-(4-chlorophenoxy)ethyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-ethoxy-3-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
6-(cyclobutylamino)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
9-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-{2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 4-{[(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazol-3-yl)formamido]methyl}benzoate
N-[2-(dimethylsulfamoyl)ethyl]-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(propan-2-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(cyclohexylmethyl)-N-[3-(4-methoxyphenyl)propyl]-6-oxopiperidine-3-carboxamide
2-cyclopentyl-N-(2-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)acetamide
4-hydroxy-N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-1-methylpiperidine-4-carboxamide
9-[2-(3-chlorophenyl)-2-hydroxyacetyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
4-hydroxy-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
1-methyl-N-{2-[4-(2-methylpropyl)morpholin-2-yl]ethyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[3-(5-methyl-2-{[2-(morpholin-4-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]ethan-1-one
1-(4-methoxybenzoyl)-4-(pyrrolidin-3-ylmethyl)piperazine
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-hydroxypyridine-3-carboxamide
1-methyl-5-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
5-(2-fluorophenoxymethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
4-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
4-methyl-2-(2-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
7-(2-methyloxane-2-carbonyl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
N,2-dimethyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(3-{4-[(3-methoxypyrrolidin-1-yl)methyl]phenoxy}propyl)morpholine
2-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}methyl)quinolin-8-ol
N-(1-carbamoylcyclopentyl)-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3,4-dihydro-2H-1-benzopyran-2-carboxamide
1-[1'-(3-acetyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
2-(3-{1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrazine
(2S,4S)-4-amino-N,N-diethyl-1-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]pyrrolidine-2-carboxamide
[(3R,4R)-1-(dimethyl-1,3-thiazole-5-carbonyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
3-methoxy-2-({[1-(3-phenylpropyl)piperidin-3-yl]amino}methyl)phenol
2-chloro-N-[(3-methyloxetan-3-yl)methyl]-5-(trifluoromethyl)benzamide
1-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}-4-(2-methylphenyl)-1,4-diazepane
3-{1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
5-[(3-fluorophenyl)methyl]-7-{[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
methyl 4-({2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}amino)benzoate
3-[(1-acetylpiperidin-4-yl)oxy]-N-[1-(4-chlorophenyl)ethyl]-4-methoxybenzamide
N-[2-(dimethylamino)ethyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(4aS,8aR)-6-[(2-fluoro-5-methoxyphenyl)methyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one