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2-(1H-indol-3-yl)-1-{4-[2-(phenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
10-methoxy-5-[5-(oxolan-2-yl)thiophene-2-carbonyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
(3S,9aR)-3-(cyclohexylmethyl)-8-(2-fluorobenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
7-fluoro-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]quinazolin-4-amine
4-{2-[(dimethylamino)methyl]phenoxy}-2-methoxypyridine-3-carbonitrile
ethyl 1-[1-(4-chlorophenyl)propan-2-yl]-4-(2-methoxyethyl)piperidine-4-carboxylate
1-{2-[(4-ethylpiperidin-1-yl)methyl]-6-methoxyphenoxy}-3-(morpholin-4-yl)propan-2-ol
1-[(2,4-difluoro-3-methoxyphenyl)methyl]-4-(2-phenoxyethyl)piperazine
3-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanamide
2-[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]-1,3-thiazole-4-carboxamide
(4aS,7aR)-1-[(3-chloro-4-fluorophenyl)methyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-{3-[1-(3-methoxypropyl)-1H-pyrazol-3-yl]phenyl}-N,N-dimethylpyrimidin-4-amine
[(3aS,6aS)-2-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
2-{2-[(2-methyl-3-oxopiperazin-1-yl)methyl]-4-(pyridin-2-yl)phenoxy}acetic acid
5-{[(propan-2-yl)(thiophen-3-ylmethyl)amino]methyl}pyrrolidin-2-one
2-{4-[(6-methoxy-2H-chromen-3-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
6-(2-butoxy-5-methylphenyl)-2-methyl-2,3-dihydropyridazin-3-one
methyl 4-[4-(3-{[2-(dimethylamino)ethyl](methyl)carbamoyl}phenoxy)piperidin-1-yl]-4-oxobutanoate
(2S)-N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}oxolane-2-carboxamide
2-{[2-(5-methylfuran-2-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
5-chloro-N-(2,2-dimethylpropyl)-N-methyl-3-phenyl-1H-indole-2-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(pyridin-4-yl)-1,4-diazepan-6-ol
3-[5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]pyridazine
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1-methyl-1H-pyrazole-4-carboxamide
(1S,5R)-3-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-(propan-2-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine-3-carboxamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(5-methylthiophen-2-yl)methyl]piperidine
(1S,5R)-3-[1-(3-chlorophenyl)piperidin-4-yl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-3-{[1-(1H-imidazole-5-carbonyl)piperidin-4-yl]oxy}-4-methoxybenzamide
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1H-pyrazole-3-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-(trifluoromethyl)benzamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
3-[2-(2,4-dimethoxy-3-methylphenyl)-1H-imidazol-1-yl]benzonitrile
1,3-dimethyl-N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}piperidin-1-yl)-1λ6-thiolane-1,1-dione
3-[(methylsulfanyl)methyl]-5-[3-(propan-2-yl)-1,2-oxazol-5-yl]-1,2,4-oxadiazole
3-butyl-4-(2,5-dimethylfuran-3-carbonyl)-1-methylpiperazin-2-one
8-(2-aminoacetyl)-3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(furan-2-ylmethyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
4-methoxy-N-({1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
8-[3-(furan-2-yl)benzoyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
2-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4H-chromen-4-one
4-fluoro-3-[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
1-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}-2-phenylethan-1-ol
(3R,5S)-1-benzyl-N3-(4-fluorophenyl)-N5-(2-methylpropyl)piperidine-3,5-dicarboxamide
4-(2-ethoxyphenyl)-3-[(4-methylpiperazin-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one