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N-(2-hydroxyethyl)-N-methyl-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)acetamide
4-[4-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenyl]but-3-yn-1-ol
1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(4aS,8aS)-2-[1-(3-methoxyphenyl)piperidin-4-yl]-decahydro-2,7-naphthyridin-4a-ol
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]pyridine-2-carboxamide
N-[3-(4-{[(2-methoxynaphthalen-1-yl)methyl]amino}piperidin-1-yl)phenyl]cyclopropanecarboxamide
{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine
3-methyl-7-[4-(piperidin-1-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
{[7-fluoro-2-(3-methoxyphenyl)quinolin-3-yl]methyl}[(4-fluorophenyl)methyl]amine
5-[1-(4-fluorophenyl)cyclopropanecarbonyl]-2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine
ethyl 1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}-3-(2-phenylethyl)piperidine-3-carboxylate
N-(3-methoxypropyl)-5-[1-(pyrimidine-5-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-(1-ethyl-1H-imidazol-2-yl)piperidine
4-{5-[(4-methylphenyl)sulfanyl]furan-2-yl}-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
4-{2-[({3-[3-(azocan-1-yl)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)amino]ethyl}phenol
4-ethyl-3-[hydroxy(phenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6-methyl-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-2-(pyrrolidin-1-yl)pyrimidin-4-amine
5-cyclobutanecarbonyl-1-[2-(dimethylamino)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[4-(1H-imidazol-2-yl)phenyl]-1H-imidazole
5-tert-butyl-4-{[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}furan-2-carboxamide
2-ethyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-methyl-1,3-thiazole-5-carboxamide
(3S,4S)-4-cyclopropyl-1-(3-methyl-1H-pyrazole-5-carbonyl)pyrrolidine-3-carboxylic acid
5-[2-(methylsulfanyl)phenoxymethyl]-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
6-(2-chlorophenyl)-N-(1-methoxypropan-2-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}[2-(2-fluorophenyl)ethyl]amine
2-(3-fluorophenyl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(1S,3R)-3-{3-[(2-methoxyphenyl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}cyclohexan-1-amine
5-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-hydroxypiperidin-4-yl)-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
N-[3-(furan-2-yl)-3-phenylpropyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
2-hydroxy-N-[1-(pyrazin-2-yl)piperidin-3-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[6-(hydroxymethyl)-1,4-oxazepane-4-carbonyl]-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
N,5-dimethyl-6-(3-phenylpiperidine-1-carbonyl)-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl){[5-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amine
4-({1-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}methyl)morpholine
1-{1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]cyclopentyl}pyrrolidine
1-{1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}piperidin-4-ol
3-{[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}-N-(1,3-thiazol-2-yl)propanamide
3-({1-[(2-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)-1-phenylurea
3-acetamido-N-(1-methyl-1H-1,3-benzodiazol-6-yl)pyrrolidine-1-carboxamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)benzamide
(3R,4S)-3,4-dimethyl-1-[3-(5-methylfuran-2-yl)benzoyl]piperidin-4-ol
(4aR,7aS)-1-(2-hydroxyethyl)-4-[2-(3-methoxyphenyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-4-ylmethyl)piperidine
(3R)-1-[(1-{[1-(4-fluoro-2-methylbenzoyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-amine
2-[4-(1-benzofuran-2-yl)phenyl]-N-methylacetamide
N-[1-(1H-1,3-benzodiazol-2-yl)-3-(methylsulfanyl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
2-{2-[(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid