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6-(2-chlorophenyl)-2-{4-[(3-hydroxypiperidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
S-[2-(furan-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-hydroxybutane-1-sulfonamido
N-ethyl-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
2-chloro-N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)pyridine-4-carboxamide
2-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-2,7-diazaspiro[4.5]decane
N-[3-(1H-pyrazol-1-yl)phenyl]-1-[(trimethylpyrazin-2-yl)methyl]piperidine-3-carboxamide
(1R,3S)-3-(2-aminoethoxy)-7-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}-7-azaspiro[3.5]nonan-1-ol
6-(quinolin-5-yl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-tert-butyl-2-[(6-ethyl-2-oxo-1,2-dihydropyridin-4-yl)formamido]acetamide
8-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(1-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
N-(propan-2-yl)-4-{[2-(thiophen-2-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3-(2-methylphenyl)pyrrolidin-3-ol
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
(4aR,8aS)-6-[(4-methoxy-3-methylphenyl)methyl]-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1-[(2,3-difluorophenyl)methyl]-4-ethyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3,5-dimethyl-1-[1-(1-methyl-1H-imidazole-2-carbonyl)pyrrolidin-3-yl]-1H-pyrazole
3-(3-fluorophenyl)-5-(thian-4-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-(thiophen-3-ylmethyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
4-(2,4-dimethyl-1,4-diazepane-1-carbonyl)-7-methyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
N-(3,3-diphenylpropyl)-2-(2-oxopyrrolidin-1-yl)propanamide
7-{pyrazolo[1,5-a]pyridine-3-carbonyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-(5-acetyl-2-methoxyphenyl)-3-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]urea
1-cyclohexyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(prop-2-en-1-yl)-1H-1,2,3-triazole-4-carboxamide
N-({1-[(3-fluoropyridin-4-yl)methyl]pyrrolidin-3-yl}methyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-butyl-3-({[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-(2-phenylethyl)-3,8-bis(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[(4-phenoxyphenyl)methyl]acetamide
[(3R,4R)-1-(3,5-dichloro-4-methylbenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
7-(1H-1,3-benzodiazole-5-carbonyl)-N-(propan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(2,5-dimethylfuran-3-carbonyl)-4-(2,6-dimethylpyridin-4-yl)piperazine
N-(1,3-dihydro-2-benzofuran-5-yl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(2-methylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-ethyl-1H-indazol-3-yl)methyl]-1H-1,2,3-triazole-5-carboxamide
(1S,5R)-6-(2-methyl-1,3-thiazole-4-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-phenyl-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-4-carbonitrile
{2-[2-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)-6-methoxyphenoxy]ethyl}dimethylamine
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-(2-methylphenyl)-1,4-diazepane
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-[(2S,4R,6R)-2-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-6-phenyloxan-4-yl]acetamide
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2,4,6-trifluorophenyl)ethan-1-one
N-[2-(pyrrolidin-1-yl)ethyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-(5-acetylthiophen-3-yl)-N-[(3-fluorophenyl)methyl]acetamide
5-(5-carbamoyl-2-methoxyphenyl)thiophene-2-carboxylic acid
(3aR,6aR)-2-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5-(pyridin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-5-(oxolan-2-yl)-N-(quinolin-5-ylmethyl)thiophene-2-carboxamide
3-(but-2-yn-1-yl)-5-[(3-fluorophenyl)methyl]-5-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
N-benzyl-5-[(2-chlorophenyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(pyridin-4-ylmethyl)-4-[6-(pyrrolidin-1-yl)pyridazin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine