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2-(4-{2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}piperazin-1-yl)pyrimidine
1-methyl-3-{[6-methyl-4-(trifluoromethyl)pyridin-2-yl]amino}pyrrolidin-2-one
1-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-methoxypiperidine
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-2,5-dimethoxybenzamide
2-(1-{[1-(4-fluoro-2-methylbenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]benzamide
3-({[(6-fluoroquinolin-2-yl)methyl]amino}methyl)-N,N-dimethylpyridin-2-amine
(3S,4R)-N-cyclohexyl-3-acetamido-4-(4-methylphenyl)pyrrolidine-1-carboxamide
2-cyclopentyl-9-[(1-ethyl-1H-pyrazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[6-hydroxy-4-(oxan-4-yl)-1,4-diazepan-1-yl]ethan-1-one
2-methyl-4-(4-{[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenyl)butan-2-ol
9-[(1-propyl-1H-imidazol-2-yl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}-N-(2-fluorophenyl)propanamide
3-{5-[2-(4,5-dimethyl-1H-pyrazol-3-yl)ethyl]-1,2,4-oxadiazol-3-yl}-6-methylpyridazine
4-ethyl-2-methyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-1,3-thiazole-5-carboxamide
N-[(1-methylpiperidin-3-yl)methyl]-3-phenyl-N-(2-phenylethyl)-1,2-oxazole-5-carboxamide
2-(2-methyl-1H-indol-3-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
1-[(2-benzyl-1,3-thiazol-4-yl)methyl]-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(dimethyl-1,2-oxazol-4-yl)acetamide
6-ethyl-2-(4-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
2-[3-(benzenesulfonyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
{1-[1-(2-methoxyethyl)piperidine-4-carbonyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-3-yl]-N-cyclopropylpropanamide
N-benzyl{[3-(pyridin-2-yl)phenyl]amino}sulfonamide
ethyl 2-[2-({1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)ethyl]-1,3-thiazole-4-carboxylate
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(dimethyl-1,3-oxazol-4-yl)methyl]-5-methylpiperidin-2-one
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetamide
(3R,4R)-4-cyclobutyl-4-hydroxy-3-methyl-N-(2-phenylethyl)piperidine-1-carboxamide
N-{5-[2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]pyridin-2-yl}cyclopropanecarboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
ethyl 3-{[3-(3-chlorobenzoyl)piperidine-1-carbonyl]amino}propanoate
N-[(5-fluoro-1H-indol-2-yl)methyl]-N,2-dimethyl-6-(piperidin-4-yl)pyrimidin-4-amine
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}thiolan-3-amine
1-[2-(cyclopent-1-en-1-yl)acetyl]-4-methanesulfonyl-1,4-diazepane-6-carboxylic acid
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-methoxyethan-1-one
2-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
[5-({[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-2-(propan-2-yloxy)phenyl]methanol
(1S,5R)-6-methanesulfonyl-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-N-[(2-methoxyphenyl)methyl]acetamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
[(2-ethylpyrimidin-4-yl)methyl](methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
1-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}azepane-2-carboxamide
methyl 6-methyl-2-(quinolin-8-yl)pyrimidine-4-carboxylate
2-(azepan-1-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
N3-cycloheptyl-4-oxo-1-(propan-2-yl)-N5-[2-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(pyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}quinolin-7-ol
4-[5-(2-methylbenzamido)-1H-pyrazol-1-yl]-N-phenylpiperidine-1-carboxamide