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[(1-cyclopentylpiperidin-4-yl)methyl]({[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl})(oxolan-2-ylmethyl)amine
3-ethyl-3-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[2-fluoro-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N-[2-hydroxy-2-(2-methylphenyl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N-{1-[1-(3-hydroxypropyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
N-cyclopropyl-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
2-(2-{1-[2-(3-fluoro-4-hydroxyphenyl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
5-cyclopropyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3,4-oxadiazol-2-amine
5-ethyl-1'-{[5-(oxan-2-yl)furan-2-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(1-cyclohexylpiperidin-3-yl)methyl][(2-methyl-1,3-thiazol-5-yl)methyl](pyridin-3-ylmethyl)amine
methyl 4-(4-{[(1-benzothiophen-2-ylmethyl)(methyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
8-(6-ethyl-2-methylpyrimidin-4-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-N-[2-(pyridin-3-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-[(2,3-dimethoxyphenyl)methyl]-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decane
4-({1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-2-yl}methyl)morpholine
1-[(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-3-yl)methyl]pyrrolidin-2-one
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-[3-(dimethylamino)-2,2-dimethylpropyl]-1H-pyrazole-4-carboxamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
2-(2,5-dimethoxyphenyl)-1-[7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
ethyl[(3-methylthiophen-2-yl)methyl](oxan-4-ylmethyl)amine
N-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-2-yl}ethyl)-2-(methylamino)acetamide
2-(4-{[2-(dimethylamino)pyrimidin-5-yl]methyl}morpholin-3-yl)-1-(thiomorpholin-4-yl)ethan-1-one
(3R,4S)-4-[ethyl({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amino]oxolan-3-ol
1-(cyclohexylmethyl)-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
1-[1-(furan-3-ylmethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-[(3S,4R)-1-(9H-fluoren-2-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-methyl-N-(quinolin-5-ylmethyl)propanamide
(2-methoxyethyl)({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)(propan-2-yl)amine
methyl 5-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-sulfonyl}-1-methyl-1H-pyrrole-2-carboxylate
2-(4-methoxypiperidine-1-carbonyl)-N-methyl-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
4-({1-[(2-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
2-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-3-methyl-1H-pyrazole-5-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(2-methoxyphenoxy)propan-2-yl]acetamide
2-[(4-methyl-1,2,5-oxadiazol-3-yl)formamido]-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)acetamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[2-(4-hydroxyphenyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(4-fluorophenyl)-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]acetamide
4-(2,6-dimethylpyridin-3-yl)-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine
5-[3-(2,3-dihydro-1H-isoindol-2-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
methyl 4-{[benzyl(oxolan-2-ylmethyl)carbamoyl]amino}-3-methylbenzoate
1-[4-(difluoromethoxy)-2-methylphenyl]-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methylurea
2-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]thiophen-3-amine
5-[(dimethylamino)methyl]-N-(5-methyl-2-pentanamidophenyl)furan-2-carboxamide
3-methyl-1-[1-(6-{[2-(pyridin-2-yl)ethyl]amino}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
1-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
3-(1H-pyrazol-5-yl)-1-[3-(pyrrolidine-1-sulfonyl)thiophene-2-carbonyl]piperidine
N-[(1-ethylpiperidin-3-yl)methyl]-N,2-dimethylthieno[2,3-d]pyrimidin-4-amine