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methyl 4-({4-[2-(2-fluorophenyl)-1-(N-methyl-1-thiophen-2-ylformamido)ethyl]piperidin-1-yl}methyl)benzoate
5-cyclobutanecarbonyl-1'-[(2-fluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-cyclopentyl-1-methyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-2-yl}pyridine
[(3-chloropyridin-4-yl)methyl](methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
7-methyl-4-(pyridin-4-yl)-6-(quinolin-4-ylmethyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
5-(7-fluoroquinazolin-4-yl)-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]pyrimidin-2-amine
3-(1-methyl-1H-pyrazol-4-yl)-N-[2-(3-phenoxyphenyl)ethyl]propanamide
N-cyclopropyl-1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-cyclopentyl-4-[4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-2-one
7-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-cyclopropanecarbonyl-8-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2S)-2-amino-2-phenyl-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-(2-methylpropyl)-5-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}piperidin-2-one
1-(2,5-dimethoxyphenyl)-3-methyl-3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]urea
N5-(1-benzothiophen-2-ylmethyl)-1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-methylquinoline
1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
1-[3-(dimethylamino)phenyl]-3-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]urea
(3R,4R)-1-(2-methanesulfonylethyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-(3-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
3-[methyl(1,3-thiazol-2-ylmethyl)amino]-1λ6-thiolane-1,1-dione
N-(2H-1,3-benzodioxol-5-yl)-5-(2-ethoxypyridin-3-yl)furan-2-carboxamide
7-cyclohexyl-2-(2-methyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
9-(2-methyl-1,3-thiazole-4-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[({[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}amino)methyl]piperidin-3-ol
6-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carbonitrile
4-[(2-fluorophenyl)methyl]-1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1,4-diazepan-5-one
3-(3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-4,5,6,7-tetrahydro-2H-indazole
5-[1-(furan-3-ylmethyl)-1H-1,2,3-triazol-4-yl]-2-methoxypyridine
1-(thiophen-3-ylmethyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
5-{[4-(oxan-4-yl)piperazin-1-yl]methyl}-1H-indole
1-(difluoromethyl)-N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-1H-pyrazole-5-carboxamide
1-{4-[(2-methoxyethyl)(methyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}[(2,3,4-trimethoxyphenyl)methyl]amine
2-[(1S,5R)-3-(6-cyanopyridine-3-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-(1,4-dioxan-2-ylmethyl)-1-(3-hydroxyphenyl)-5-oxopyrrolidine-3-carboxamide
2-(2,2-dimethylpropanoyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(3R,4R)-4-(hydroxymethyl)-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidin-3-ol
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
N-tert-butyl-4-{3-[(pyridin-3-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
2-[2-(furan-2-yl)azepane-1-carbonyl]quinoline
5-({2-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1-methyl-1H-1,2,3,4-tetrazole
(4aS,7aR)-4-[(dimethylcarbamoyl)methyl]-6,6-dioxo-N-pentyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-{5-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-ylmethyl]furan-2-yl}benzonitrile
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(2,5-dimethylfuran-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-methyl-5-{[2-(naphthalen-2-yloxy)propanamido]methyl}-1,2,4-oxadiazole-3-carboxamide
8-(3-hydroxypyridine-2-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid