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N-[3-(4-chlorophenoxy)-2-hydroxypropyl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
4-[2-(2-chlorophenyl)ethyl]-11-{methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
4-ethyl-3-(1-{2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(morpholin-4-yl)-1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole
2-({2-[methyl(quinoxalin-2-ylmethyl)carbamoyl]phenyl}amino)acetic acid
N-cyclopropyl-3-{[(2,3-dihydroxypropyl)(methyl)carbamoyl]amino}-4-methoxybenzamide
3-hydroxy-5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
2-[4-(diphenylmethyl)piperazine-1-carbonyl]morpholine
4,6-dimethyl-1-(3-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}-3-oxopropyl)-1,2-dihydropyrimidin-2-one
(4aS,8aR)-1-(2-aminoethyl)-N-[(4-fluorophenyl)methyl]-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
4-[4-({[2-fluoro-4-(trifluoromethyl)phenyl]methyl}amino)piperidin-1-yl]-6-methylpyrimidin-2-amine
2-{4-[2-(methoxycarbonyl)thiophene-3-sulfonamido]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
5-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2-(propan-2-yl)pyrimidine
4-(1-methyl-1H-pyrazol-4-yl)-N-[3-(pyridin-2-yl)propyl]pyrimidin-2-amine
5-[1-(2-hydroxyethyl)-3-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
5-butyl-1-(3-chlorophenyl)-4-(3-methyl-1H-pyrazole-5-carbonyl)piperazin-2-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(6-hydroxypyrimidin-4-yl)methyl]-5-methylpiperidin-2-one
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
3-(propan-2-yloxy)-6-{3-[1-(1,3-thiazol-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridazine
(3S,4R)-N-benzyl-3-(dimethylamino)-N-methyl-4-(propan-2-yl)pyrrolidine-1-sulfonamide
7-methyl-2-[1-(4-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
(5S,9aS,9bS)-5-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-{2-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
3,5-dimethyl-N-[2-(1-methylpiperidin-4-yl)ethyl]adamantane-1-carboxamide
2-cyclopentyl-4-{4-[2-(2-methoxyphenyl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2-methylprop-2-en-1-yl)-1H-pyrazole-3-carboxamide
2-(2-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
(1,3-benzothiazol-2-ylmethyl)({[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
2-[2-(dimethylamino)ethyl]-9-(3-methoxypyrazin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-(pyridine-2-carbonyl)-7-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-ethyl-2-(furan-2-yl)-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-oxoacetamide
2-[2-methoxy-5-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)phenoxy]acetic acid
6-{1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}pyrimidin-4-ol
ethyl 1-(2-methoxyethyl)-5-(naphthalene-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-[(3-methoxyphenyl)sulfanyl]acetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(4-methyl-1,3-thiazol-2-yl)-1,4-diazepane
4-methyl-2-[4-(pyridin-4-ylmethyl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
(1S,6R)-9-[3-(1,2-oxazinan-2-yl)propanoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(3S)-2-oxoazepan-3-yl]benzamide
(1r,4r)-4-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)cyclohexan-1-ol
6-methyl-2-[1-(5-methylthiophene-3-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
4-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)piperazine-1-carboxamide
(2S)-4,4-difluoro-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}pyrrolidine-2-carboxamide
1-(3,5-dimethylphenyl)-4-[(3-ethoxy-4-hydroxyphenyl)methyl]piperazin-2-one
2-methoxy-1-[1'-(2-methyl-6-propylpyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
3-(2H-1,3-benzodioxol-5-yl)-5-(ethanesulfonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
5-acetyl-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]thiophene-3-carboxamide
3-ethyl-8-(2-methyl-4-phenylpyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one