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N-(2-hydroxyethyl)-4-(1H-pyrazol-3-yl)-N-(1,3-thiazol-2-ylmethyl)benzamide
3,5-dimethyl-2-({[4-(pyridin-2-yl)pyrimidin-2-yl]amino}methyl)pyridin-4-ol
2-(2-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}ethyl)pyridine
6-cyano-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyridine-3-carboxamide
1-(2-{1-[1-(4,6,7-trimethylquinazolin-2-yl)piperidin-4-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-{[2-(2-methyl-1,3-thiazol-4-yl)acetamido]methyl}benzoate
4-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-{[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-4-methoxy-3,5-dimethylpyridine
8-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2,4-dimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)quinoline-7-carboxamide
4-chloro-2-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]-1H-indole
1-(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidin-1-yl)-2-ethoxyethan-1-one
4-{1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}benzoic acid
(1S,3R)-N-[3-(furan-2-yl)propyl]-3-[2-(methylsulfanyl)acetamido]cyclopentane-1-carboxamide
N,3,5-trimethyl-N-[1-(pyrimidin-4-yl)ethyl]-1H-indole-2-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-[3-(piperidine-1-carbonyl)phenyl]urea
N-(2-methoxyethyl)-3-{[1-(thian-4-yl)piperidin-4-yl]oxy}benzamide
(1R,5S)-6-methyl-7-oxo-N-[3-(2-oxopyrrolidin-1-yl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[3-(1H-indol-1-yl)propyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
2-amino-4-(2,1,3-benzothiadiazol-5-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)pyrrolidine-3-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-[(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]benzamide
5-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}-2-methoxyphenol
N-methyl-N'-(4-methylphenyl)-N-[2-(oxan-4-yl)ethyl]propanediamide
3,5-dimethyl-4-{[2-(3-phenylpropyl)morpholin-4-yl]methyl}phenol
2,7-dioxo-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,3-diazepane-4-carboxamide
2-cyclopropyl-8-(5,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
methyl({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
6-methyl-4-oxo-N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-4H-pyran-2-carboxamide
2-oxo-N-[(2-phenoxypyridin-3-yl)methyl]-1,2-dihydroquinoline-4-carboxamide
4-(1H-indol-3-yl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]butan-1-one
N-[(4-methanesulfonylphenyl)methyl]-N-methylthian-4-amine
2-(1-benzyl-4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl)ethan-1-ol
5-methyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]benzamide
5-[2-(morpholin-4-ylmethyl)phenyl]-1H-indazol-3-amine
4-(2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzoyl)thiomorpholine
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(2-phenoxyethoxy)phenyl]propanamide
(2S)-2-amino-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
2-methyl-7-{[5-(1,2-oxazol-5-yl)furan-2-yl]sulfonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-amino-6-tert-butyl-4-(3,4,5-trimethoxyphenyl)pyridine-3-carbonitrile
4-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-methyl-1H-pyrazole
11-(pentan-2-yl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
[(2S,6S)-4-(5-methyl-1,2-oxazole-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
(1S,5R)-3-[2-(4-methylphenyl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(trifluoromethyl)-4-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}morpholine
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
N,6-dimethyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyridazin-3-amine