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3-methyl-1-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]butan-1-ol
2-methyl-4-{3-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]phenyl}butan-2-ol
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
5-hydroxy-N-{2-[(pyridin-2-ylmethyl)carbamoyl]phenyl}pyrazine-2-carboxamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-methyl-N-(3-methylbutyl)piperidine-4-carboxamide
1-tert-butyl-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-pyrrole-3-carboxamide
1-cyclohexyl-3-(cyclopropylmethyl)-5-(1,4-diazepane-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
5-{1-[(2,4-dimethylphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
(2S,4R)-1-benzyl-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
1-(1-ethylpiperidine-2-carbonyl)-4-phenylpiperidine-4-carbonitrile
4-(2-amino-6-methylpyrimidin-4-yl)-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-methyl-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
1'-cyclohexanecarbonyl-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-methyl-8-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-methylpropanamide
N-[2-(diethylamino)ethyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
4-hydroxy-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-phenylpyrimidine-5-carboxamide
ethyl 3-benzyl-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-3-carboxylate
2-(2-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-methoxy-4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl})amine
2-(3-{4-[1-(morpholin-4-yl)ethyl]phenyl}phenoxy)acetamide
1-benzyl-N3-[(5-chlorothiophen-2-yl)methyl]-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(2-methylpropyl)-7-(methylsulfanyl)-3-({[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
(4aR,7aS)-1-(2-methoxyethyl)-4-(3-methoxypropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-phenyl-1H-pyrazole-4-carboxamide
2-cyclopentyl-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1-methyl-1H-1,2,3-benzotriazole-5-carboxamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
1,5-dimethyl-N-[1-(morpholin-4-ylmethyl)cyclopentyl]-1H-pyrrole-2-carboxamide
N-(1-hydroxybutan-2-yl)-2-(methylamino)-N-(pyridin-2-ylmethyl)benzamide
4-(2,6-dimethylpyridin-3-yl)-2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}pyrimidine
5-methoxy-2-({3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
5-{1-[(4-fluorophenyl)methyl]pyrrolidin-2-yl}-N-[2-(1H-imidazol-4-yl)ethyl]thiophene-2-carboxamide
N-[3-(4-{[1-(1H-indol-1-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]ethane-1-sulfonamide
1-methyl-3-{[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-methyl-1-benzofuran-5-carboxamide
2-(3-fluorophenyl)-N-(3-hydroxy-3-phenylpropyl)-N-methyl-1,3-benzoxazole-5-carboxamide
1-{4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenyl}-2-(morpholin-4-yl)ethan-1-ol
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-[6-oxo-4-(piperazin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
2,8-dimethyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)quinoline-4-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
methyl 1-methyl-2-[3-(pyridin-3-yl)azetidin-1-yl]-1H-1,3-benzodiazole-5-carboxylate
2-(5-fluoro-2-methoxyphenyl)-3-(pyrrolidine-1-carbonyl)pyridine
2-methoxy-4-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}pyridine-3-carbonitrile