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1-[2-(thiophen-3-yl)pyrimidin-4-yl]pyrrolidin-3-ol
5-acetyl-6-methyl-3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2,2-difluoro-N-[(1-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}piperidin-3-yl)methyl]acetamide
5-chloro-4-({[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amino}methyl)-2-methoxyphenol
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-(1,2-oxazol-3-ylmethyl)acetamide
1-{2-[(6-cyclopropylpyrimidin-4-yl)amino]ethyl}imidazolidin-2-one
N-[(3S,4R)-1-{2-[4-(dimethylamino)phenyl]acetyl}-4-propylpyrrolidin-3-yl]acetamide
2-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]pyridine-4-carboxamide
[(3R,4R)-1-cyclobutanecarbonyl-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
4-{2-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-2-yl]ethyl}phenol
5-[3-(4-methylpiperidine-1-carbonyl)phenyl]-1H-indazol-3-amine
2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-3,5-dimethyl-1H-indole
(2S)-N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}oxolane-2-carboxamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)amine
2,4-dimethoxy-N-(oxolan-3-yl)benzamide
methyl[(4-methylphenyl)methyl]{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-(furan-3-ylmethyl)-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})[(6-methylpyridin-2-yl)methyl]amine
1-(3-chlorophenyl)-4-[(3-{2-[1-(1,3-thiazole-5-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine
methyl(oxan-2-ylmethyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
1-[2-(2,5-dimethyl-1H-pyrrol-1-yl)ethyl]-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperazine
ethyl 4-[1-(pyridin-2-ylmethyl)piperidin-3-yl]piperazine-1-carboxylate
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2,3-dimethyl-1H-indole-5-carboxamide
5-methyl-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-2-(thiophen-3-yl)-1,3-oxazole
2-(4-{[methyl(1-phenylpropyl)amino]methyl}phenyl)-3H,4H,5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-one
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}propane-1-sulfonamide
3-(benzylsulfanyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]propan-1-one
2-ethoxy-4-({3-[(3-fluorophenyl)amino]piperidin-1-yl}methyl)phenol
{1-ethyl-5-[4-(1H-pyrazol-3-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
5-({[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-(quinolin-5-yl)piperidine-1-carboxamide
5-{[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-N,N-dimethylfuran-2-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-3-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}benzamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(cyclopropanesulfonyl)piperidin-3-ol
1-(1-acetylpiperidin-4-yl)-N-[4-(3-fluorophenyl)phenyl]pyrrolidine-2-carboxamide
1-[4-(1,3-benzoxazol-2-yl)-1,4-diazepan-1-yl]-2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({[(3-methylphenyl)methyl]amino}methyl)piperidin-2-one
2-[2-chloro-4-({methyl[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]acetamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}pyridine-3-carboxamide
methyl 1-(2-methylpropyl)-5-[(pentan-3-yl)amino]-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(morpholine-4-carbonyl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[2-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethyl]pyrrolidin-2-one
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}thian-4-amine
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1-(pyridin-2-yl)piperidine-3-carboxamide
(1S,4S)-5-[5-(4-methoxyphenyl)furan-2-carbonyl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
11-methyl-5-[2-(methylsulfanyl)ethyl]-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
2-{4-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carbonyl]morpholin-3-yl}acetic acid
2-[(2-fluorophenyl)methyl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,3-benzoxazole-6-carboxamide