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1-[(3,5-difluorophenyl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
4-[(diethylamino)methyl]-5-ethyl-N-methyl-N-(prop-2-yn-1-yl)furan-2-carboxamide
N-(3-fluorophenyl)-1-(thiophene-3-carbonyl)piperidin-3-amine
5-[(3E)-pent-3-enoyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetamide
3-(2-phenylethyl)-5-[(1R,2S,3S,4R,5S)-tricyclo[3.2.1.02,4]octan-3-yl]-1H-1,2,4-triazole
2-methyl-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-pyrrol-1-yl)propan-1-one
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-[(2-ethylpyrimidin-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
2-benzyl-9-[(3-fluoro-5-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(2-fluorophenoxymethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,3-oxazole-4-carboxamide
5-(1H-pyrazol-1-ylmethyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]furan-2-carboxamide
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({2-methyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}methyl)piperidin-2-one
3-{[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-1-yl]methyl}phenol
2-{5-[(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-(4-chlorophenyl)-4-[2-(3-hydroxypiperidin-1-yl)-2-oxoethyl]-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1,4-oxazepan-6-ylmethyl)-5-(trifluoromethyl)pyridin-2-amine
2-(propan-2-yl)-8-(5-propylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
2,5,6-trimethyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}pyrimidin-4-amine
N-[(2,4-dihydroxyphenyl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
5-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-cyclopentyl-2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)propanamide
1-(2-{[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl](methyl)amino}ethyl)piperidin-2-one
(1S,5R)-6-(5-propylthiophene-3-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
{1-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
7-(cyclobutylmethyl)-2-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
4-(1H-pyrazol-1-ylmethyl)-N-{3-[(trifluoromethyl)sulfanyl]phenyl}piperidine-1-carboxamide
1-(2-methylphenyl)-4-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperazin-2-one
2-amino-4-[2-(ethylamino)pyrimidin-5-yl]-6-(2-methylbutan-2-yl)pyridine-3-carbonitrile
5-[1-(4-fluorobenzoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
(4aR,8aS)-1-(cyclohexylmethyl)-6-[(2,6-difluorophenyl)methyl]-decahydro-1,6-naphthyridin-2-one
N-(2-methoxyethyl)-1-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)piperidine-3-carboxamide
2-[(3,4-difluorophenyl)methyl]-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-[3-(4-benzyl-4-hydroxypiperidine-1-carbonyl)piperidin-1-yl]acetamide
1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazole
3-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1H-pyrazole
4-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}pyrrolidin-2-one
N-methyl-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
4-(4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)piperidin-4-ol
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2-methylpyrimidine-5-carboxamide
3-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-ethyl-1-(pyridin-4-ylmethyl)urea
2-{4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenoxy}ethan-1-ol
6-{2-cyclopentyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-(1-methylpiperidin-4-yl)-3-[2-(methylsulfanyl)benzoyl]piperidine
3,6-dimethyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
1,5-dimethyl-4-{[3-(4-methylphenoxymethyl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
1-{5-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
4-{4-[3-(hydroxymethyl)-4-methylpiperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol