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4-(2-methyl-1H-imidazol-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]aniline
4-{6-[3-(propan-2-yloxy)phenyl]pyridazin-3-yl}thiomorpholine
methyl 3-{[(2-methoxyphenyl)formamido]methyl}-5-(pyrazine-2-amido)benzoate
4-(5-chloro-2-fluorobenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-1-[3-(1H-imidazol-1-yl)propyl]urea
5,5-dimethyl-3-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-oxazolidine-2,4-dione
4-ethyl-3-(piperidin-4-ylmethyl)-1-(quinolin-8-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
9-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)-N-(propan-2-yl)pyridine-2-carboxamide
7-chloro-4-[1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-cyclopropyl-5-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
2-[1-(1,3-thiazol-5-yl)propan-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
(2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-4-yl)methanol
2-(2-oxopyrrolidin-1-yl)-N-[2-(2-phenoxyethoxy)phenyl]propanamide
3-(2-hydroxyethyl)-1-(5,6,7,8-tetrahydronaphthalen-1-yl)-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
N-methyl-2-{3-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}carbamoyl)amino]phenyl}acetamide
3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-8-(pyrimidin-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
1-cyclopentanecarbonyl-N-[2-(pyridin-4-yl)ethyl]piperidine-4-carboxamide
(1R,5R)-3-(2-methyl-1H-pyrrole-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
1-[4-(1H-pyrazol-1-yl)phenyl]-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]piperidin-4-amine
2-[1-(furan-2-ylmethyl)-4-{[1-(propan-2-yl)piperidin-4-yl]methyl}piperazin-2-yl]ethan-1-ol
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
3-({4-[1-(cyclopentylmethyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-{methyl[(4-methylphenyl)methyl]amino}ethan-1-one
3-(furan-2-yl)-1-[3-(2-phenylacetyl)piperidin-1-yl]propan-1-one
(3aR,5S,6S,7aS)-2-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)-octahydro-1H-isoindole-5,6-diol
8-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-(4-methoxy-2-methylphenyl)pyridine-2-carbonitrile
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-amino-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-6-(propan-2-yl)pyrimidine-4-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(4-methyl-1H-imidazol-2-yl)methyl]piperazine
1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-3-yloxy)ethan-1-one
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]acetamide
1-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]-3-{1-oxaspiro[4.4]nonan-3-yl}urea
({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[2-(2-methylphenyl)pyrimidin-5-yl]methyl}amine
1-butyl-4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
(3E)-N-(3-hydroxypropyl)-N-[(5-methylthiophen-2-yl)methyl]pent-3-enamide
5-[methyl(1,2-oxazol-5-ylmethyl)amino]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
7-(2-methoxyethyl)-2-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decane
N-(1-benzylpyrrolidin-3-yl)-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-(2-hydroxyphenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
5-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidine
N-(3-{3-methyl-3,9-diazaspiro[5.6]dodecane-9-carbonyl}phenyl)acetamide
3-[2-(3,4-difluorophenyl)ethyl]-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
methyl 6-({cyclopropyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-3-(oxolane-2-amido)thieno[2,3-b]pyridine-2-carboxylate
[(1S,3S,3aS,6aR)-3-(3-ethenylphenyl)-5-methyl-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
1-[cyclohexyl(methyl)amino]-3-[4-({[(2,3-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
4-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]azepane