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1-(1-methyl-1H-pyrrol-2-yl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethane-1,2-dione
1-butyl-4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidine
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
(1S,5R)-3-[(4-methoxy-2,5-dimethylphenyl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-6-methylpyridine-3-carbonitrile
4-[cyclohexyl(methyl)amino]-4-[1-(propan-2-yl)piperidin-4-yl]but-2-yn-1-ol
4-(1-{1-[(3-phenoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
1-ethyl-5-(1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-phenyl-1H-imidazol-5-yl)-1H-1,2,4-triazole
ethyl 4-[5-(3-chlorophenyl)-1,2,4-triazin-3-yl]piperazine-1-carboxylate
4-{4-[(2-hydroxyethyl)sulfanyl]benzoyl}-1-(4-methylphenyl)piperazin-2-one
7-(5-chloropyridine-2-carbonyl)-N,N-dimethyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[5-(methoxymethyl)furan-2-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-methyl-4-[4-({[(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amino}methyl)phenyl]but-3-yn-2-ol
N-{2-[(1R,7S)-6-(azepane-1-carbonyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-3-yl]ethyl}acetamide
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
2-{[(1S,5R)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzoic acid
1-(2,1,3-benzoxadiazol-5-ylmethyl)-3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-methylurea
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]propan-1-one
ethyl 4-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-amido}piperidine-1-carboxylate
5-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-(5-methylfuran-2-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
4-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-methoxypyridine-3-carbonitrile
N-methyl-N-[(4-methylphenyl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
5-(3-ethyl-1-methyl-1H-pyrazol-5-yl)-3-(oxolan-2-ylmethyl)-1,2,4-oxadiazole
3-[4-(2-chlorophenyl)-4H-1,2,4-triazol-3-yl]-1-methylpiperidine
ethyl 1-{2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperidine-3-carboxylate
(3aS,6aS)-2-cyclopropanecarbonyl-5-(5-propyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-(2,3-dihydro-1H-inden-1-yl)-N-methylacetamide
N-[4-(1-ethyl-1H-1,2,4-triazol-5-yl)-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-2-methylpropanamide
1-(cyclohexylmethyl)-3-[(4-ethylpiperazin-1-yl)methyl]-3-hydroxypiperidin-2-one
N2-benzyl-6-(1H-pyrazol-4-yl)-1,3,5-triazine-2,4-diamine
2-cyclopentyl-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)acetamide
{2-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1,3-thiazol-4-yl}methanol
3-{[2-(1H-imidazol-1-yl)ethyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(3-methylphenyl)piperidine
5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[(2-fluorophenyl)methyl]piperidin-2-one
N-(3-ethoxypropyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-ethyl-2,5-dimethyl-1H-pyrrole-3-carboxamide
N-(furan-2-ylmethyl)-N,1-dimethyl-5-{[3-(methylsulfanyl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-propyl-1,4-diazepane
8-(3,4,7-trimethyl-1H-indole-2-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
3-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)phenol
N,2,7,8-tetramethyl-N-[2-(1H-pyrazol-4-yl)ethyl]quinoline-4-carboxamide
3-(1-butyl-1H-imidazol-2-yl)-1-(4-fluoro-3-methoxybenzoyl)piperidine
(3S,4S)-4-methoxy-N-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidin-3-amine
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-4-(piperidin-3-yl)benzamide
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-(4-fluorophenyl)-1-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-1,2,3,6-tetrahydropyridine