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3-[2-(dimethylamino)ethyl]-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(oxolan-2-ylmethyl)urea
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-methyl-1,2,3,6-tetrahydropyridine
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-5-methylthiophene-2-carboxamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][(4-phenyl-1,3-thiazol-5-yl)methyl]amine
1-(3-{[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amino]methyl}phenyl)ethan-1-one
2-(methylamino)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
2-{3-methyl-4-[2-(methylsulfanyl)ethyl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl}acetic acid
methyl 4-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}benzoate
N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(pyrrolidin-1-yl)benzamide
1-(1-{[2-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
1-propyl-5-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl]piperidin-2-one
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-N-[(4-fluorophenyl)methyl]piperidine-1-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-{[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]amino}pyrrolidin-2-one
2-{4-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]piperazin-1-yl}pyridine-3-carbonitrile
1-(carbamoylmethyl)-N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-4-carboxamide
2-{4-[3-(2-methoxyphenoxy)propyl]phenyl}-1,3,4-oxadiazole
14-(3-methyl-1-benzothiophen-2-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1-(1,2,4-oxadiazol-3-ylmethyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-methyl-N-(quinolin-8-ylmethyl)acetamide
2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-1,3-thiazole-4-carboxamide
5-(dimethylamino)-2-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,3-dihydropyridazin-3-one
5-acetyl-N-[(4-methanesulfonylmorpholin-2-yl)methyl]thiophene-3-carboxamide
methyl 2-{3-[(phenylformamido)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}benzoate
8-[(4-hydroxyphenyl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(2-fluorophenoxy)-1-(2-propoxyacetyl)piperidine-4-carboxylic acid
methyl (2S,4R)-4-hydroxy-1-({4-[(4-methylpyridin-3-yl)carbamoyl]phenyl}methyl)pyrrolidine-2-carboxylate
3-{[4-(3,4-dimethoxyphenyl)-1H-1,2,3-triazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
(2S,4S)-4-amino-1-{3-[5-(thiophen-2-yl)furan-2-yl]propanoyl}pyrrolidine-2-carboxylic acid
N,2,8-trimethyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}quinoline-4-carboxamide
1-[({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]cyclopentane-1-carboxamide
1-[(2S)-2-[4-(2-phenylpyrimidin-4-yl)piperidine-1-carbonyl]pyrrolidin-1-yl]ethan-1-one
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(2-hydroxyphenoxy)acetamide
2-[1-(cyclohexylmethyl)-4-{[5-(hydroxymethyl)furan-2-yl]methyl}piperazin-2-yl]ethan-1-ol
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carboxamide
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
N-cyclopentyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-(3-phenylprop-2-yn-1-yl)acetamide
5,6-dimethyl-1-{[3-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-1,3-benzodiazole
1-(1-benzofuran-2-ylmethyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
5-[4-(2-phenylethyl)piperidine-1-carbonyl]-2-(thiophen-3-yl)pyridine
2-[8-benzyl-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
5-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-1-methylpiperidin-2-one
1-[5-(oxolan-2-yl)thiophene-2-carbonyl]-4-(thian-4-yl)piperazine
2-methoxy-5-{[(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amino]methyl}phenol
5-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methyl-1H-1,3-benzodiazole
3-cyclohexyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-pyrazole-4-carboxamide
4-[8-methyl-3-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)quinolin-2-yl]piperazin-2-one
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-2-[methyl(pyridin-2-ylmethyl)amino]acetamide