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(3aS,6aS)-2-cyclopropanecarbonyl-5-(trimethyl-1H-pyrazole-4-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[2-(1-benzoylpiperidin-2-yl)ethyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
5-{[(2-methoxynaphthalen-1-yl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(3-chloro-4-methoxyphenyl)-4-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}pyrrolidin-2-one
2-[5-(2,3,4,9-tetrahydro-1H-carbazole-1-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
3-{[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]methyl}-1-(2-chloroprop-2-en-1-yl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
9-(3-hydroxy-2-methylbenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(piperazine-1-carbonyl)benzene-1-sulfonamide
5-[4-(4-acetylphenyl)piperazin-1-yl]-N-benzyl-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-[2-(aminomethyl)-4-fluoro-2,3-dihydro-1-benzofuran-7-yl]-N,N-diethylfuran-2-carboxamide
6-cyclopropyl-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine
ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](3-phenylbutyl)amine
5-cyano-2-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
2-[4-(1-benzyl-1H-pyrazol-4-yl)phenyl]-N-methylacetamide
3-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}phenol
1-cycloheptanecarbonyl-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
4-(4-fluorophenoxy)-1-(3-methylfuran-2-carbonyl)piperidine-4-carboxylic acid
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-cyclopropyl-1-(2-{1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
[(3R,4S)-1-[(6-chloroquinolin-2-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
3-chloro-6-(pyrimidin-5-yl)pyridine-2-carboxylic acid
2-{4-[4-(1-methoxyethyl)phenyl]phenyl}-N-methylacetamide
3-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]-N-(thiophen-2-ylmethyl)aniline
N-benzyl-N-methyl-3-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}propanamide
2-[(3,4-difluorophenyl)methyl]-8-(pyrimidin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
7-[(3,4-difluorophenyl)methyl]-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
(1,3-benzothiazol-2-ylmethyl)({[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
2-(3-phenylpropyl)-4-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]morpholine
N-cyclopentyl-N-[(2-methoxyphenyl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
2-cyclobutanecarbonyl-7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
1-[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-cyclopentanecarbonyl-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-ethyl-2,4-dimethyl-6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-(1,2-oxazol-3-ylmethyl)-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
9-(2-hydroxy-4-methylpentanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2-methoxyethyl)-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(3-methylthiophen-2-yl)methyl]propanamide
2-[5-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
3,5-difluoro-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]pyridine-2-carboxamide
N-ethyl-2-(4-fluorophenyl)-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}benzamide
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-(pyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N,N-diethyl-5-methyl-3-(1-methylpiperidin-4-yl)-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclopentanamine
6-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]-N,N-dimethylpyrazin-2-amine
6-({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}amino)pyridine-3-carboxamide
4-[(2-fluorophenyl)methyl]-11-{[2-(pyridin-3-yl)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[3-(piperidin-1-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-(1-methyl-1H-pyrazol-4-yl)-1-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}propan-1-one
8-benzyl-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione