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1-{1-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]azetidin-3-yl}piperidine
9-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(3-{[4-(2-ethylphenyl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)-1H-1,2,3,4-tetrazole
N-[2-(1-ethylpiperidin-3-yl)ethyl]-2-methoxybenzene-1-sulfonamide
(3S,4R)-1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-4-(hydroxymethyl)piperidin-3-ol
2-benzyl-9-(oxan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(1-{[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}pyrrolidin-3-yl)methanamine
N-[(2-methoxyphenyl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(2-chloro-4-fluorophenyl)-N-methyl-N-(quinolin-5-ylmethyl)acetamide
2-[2-(dimethylamino)ethyl]-8-(trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-(methylsulfanyl)-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
N-ethyl-4-(3-hydroxy-3-methylbutyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)cyclopent-3-ene-1-carboxamide
N,3,6-trimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
(4aS,8aR)-6-(ethanesulfonyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(dimethylamino)ethyl]-2-methyl-N-{[8-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}propanamide
2-{[(2,5-dimethylphenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
4-methyl-2-(4-methylpiperazin-1-yl)-5-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]pyrimidine
1-{4-[({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)methyl]phenyl}pyrrolidin-2-one
2-{[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]methyl}-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
2-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-7-(4-fluorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
4-[(3-chloropyridin-4-yl)methyl]-2-(piperidin-1-ylmethyl)-1,4-oxazepane
4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-N-(pyridin-4-ylmethyl)pyrimidin-2-amine
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-{[1-(morpholin-4-yl)cycloheptyl]methyl}urea
[(1-ethylpyrrolidin-3-yl)methyl](1H-indol-7-ylmethyl)methylamine
7-(2-methylphenyl)-4-(3-methylpyridine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2-cyclopentyl-2-phenylacetyl)-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(piperidin-4-ylmethyl)benzamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}cyclopentanamine
4-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-ol
N-methyl-N-[2-(oxan-2-yl)ethyl]-2-(phenylsulfanyl)acetamide
3-{2-oxo-2-[1-(pyridin-2-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl]ethyl}-3,4-dihydroquinazolin-4-one
2-methylpropyl N-{[(3S,4S)-3-hydroxy-1-(3-methylfuran-2-carbonyl)piperidin-4-yl]methyl}carbamate
2-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-3,4-dihydroquinazolin-4-one
7-(cyclobutylmethyl)-2-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-[(2E)-3-phenylprop-2-en-1-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[(3R,4R)-3-hydroxy-1-{2-[(trifluoromethyl)sulfanyl]acetyl}piperidin-4-yl]pyridine-2-carboxamide
1-(cyclohexylmethyl)-N,N-dimethyl-5-(piperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(2-aminoethyl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-(1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-yl)acetamide
N-(2H-1,3-benzodioxol-5-yl)-3-{[ethyl(oxan-4-yl)amino]methyl}benzamide
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(3-methylphenoxy)azetidine
2-[(2-{[2-(diethylamino)ethyl](methyl)carbamoyl}phenyl)amino]acetic acid
(2R)-1-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]propan-2-ol
2-(4-{[3-(cyclopentyloxy)phenyl]methyl}piperazin-1-yl)-N-ethylacetamide
N-[2-(4-ethylmorpholin-2-yl)ethyl]-2-(2,3,4-trifluorophenyl)acetamide
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-2-(2-methoxyphenoxy)-2-methylpropan-1-one
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-oxazole-4-carbonyl)piperidine