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2-cyclobutyl-N-[(3R,4S)-4-(propan-2-yl)-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]acetamide
4-methoxy-6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidine
4-{4-[3-(dimethylamino)pyrrolidin-1-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]furan-3-carboxamide
3-ethyl-8-(8-hydroxy-5,7-dimethylquinoline-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2,5-dioxoimidazolidin-1-yl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
(4aS,8aR)-6-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-5,6-dimethylpyrimidine
1-(3,5-dimethoxybenzoyl)-N-(thiolan-3-yl)piperidine-4-carboxamide
N-cyclopropyl-7-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-amine
4-(1-benzofuran-2-yl)-6-methylpyrimidin-2-amine
1-methyl-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-(adamantan-2-ylmethyl)-6-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(3-chloro-1-benzothiophen-2-yl)methyl]-1-cyclopropyl-6-oxopiperidine-3-carboxamide
2-[2-(4-phenyl-1H-imidazol-5-yl)phenoxy]acetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(4-methyl-2-oxo-1,2-dihydroquinolin-1-yl)acetamide
[(4,5-dimethylfuran-2-yl)methyl]({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
[1-(azepan-1-yl)propan-2-yl][(4-ethyl-1,3-thiazol-2-yl)methyl]amine
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-(propylsulfanyl)ethan-1-one
5-cyclopropanecarbonyl-1'-(3-propyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2-methylpyrrolidin-1-yl)-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridine
5-(1,3-benzothiazol-2-ylmethyl)-N-cyclopentyl-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-3-methylpiperidine
4,6-dimethyl-N-(3-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methoxy}phenyl)pyrimidin-2-amine
2-(dimethylamino)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
5-benzyl-5-(3-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-[3-(4-fluorophenoxy)azetidine-1-carbonyl]-3,5,7-trimethyl-1H-indole
(3R,4R)-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-5-methylthiophene-2-carboxamide
2-methoxy-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-{2-[(4aS,8aR)-1-(3-methylbutyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
1-[(4-methyl-5-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]azepane
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]-2,4-dimethyl-3-oxopiperazine-1-carboxamide
(3R,4R)-4-ethyl-1-(2-methyl-1,3-benzothiazole-5-carbonyl)piperidine-3,4-diol
(2S,4R)-1-(5-chloro-2-methylbenzoyl)-4-(dimethylamino)pyrrolidine-2-carboxylic acid
8-(6-aminopyrimidin-4-yl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N-cyclopropyl-3-(1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}piperidin-3-yl)propanamide
N-{1-[7-(2,2-diphenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-methoxypropanamide
7-(2-cyclohexylethyl)-2-[2-(methylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-7-methoxy-6-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
(2S,4S,5R)-5-(4-chlorophenyl)-4-(4-hydroxypiperidine-1-carbonyl)-1,2-dimethylpyrrolidine-2-carboxylic acid
N-({1-[(4-methoxy-3-methylphenyl)methyl]pyrrolidin-3-yl}methyl)cyclobutanecarboxamide
6-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pyridine-2-carboxamide
N-(6-fluoropyridin-3-yl)-4-[(1-methylpiperidin-3-yl)methyl]piperazine-1-carboxamide
8-{[4-(2-methylpropyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2,1,3-benzoxadiazol-5-ylmethyl)[(5-tert-butyl-1H-pyrazol-3-yl)methyl]methylamine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,3,4,7-tetramethyl-1H-indole-2-carboxamide