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3-(2-{[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
3-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)sulfamoyl}-N,N-dimethylbenzamide
3-acetamido-N-[(2-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)benzamide
2-cyclopropyl-6-{[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]methyl}pyrimidin-4-ol
1-(2-methoxy-5-{[(2-methylpropyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
3,5-dimethoxy-N-{[1-(pyrimidin-2-ylmethyl)piperidin-3-yl]methyl}benzamide
{3-[5-(3-fluoropyridin-4-yl)-1,2,4-oxadiazol-3-yl]phenyl}methanol
2-{4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-3-carboxamide
N-methyl-2-[methyl({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl})amino]acetamide
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-5-methyl-2-phenyl-1H-imidazole-4-carboxamide
N-({5-[(2,5-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-(2-hydroxyethyl)-2,3-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]quinoxaline-6-carboxamide
{1-[(dimethyl-1,3-thiazol-2-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
ethyl 2-(3-{[2-(propan-2-yl)phenyl]carbamoyl}propanamido)propanoate
4-{[4-(cyclopentyloxy)phenyl]methyl}-1,4-oxazepan-6-ol
1-[3-(3-ethylphenoxy)azetidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
N-[(1-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)methyl]acetamide
1-(2,3-dimethyl-1H-indole-5-carbonyl)-4-(4-fluorophenyl)piperidin-4-ol
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(3-phenylbutyl)piperidine
3-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}phenol
N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-(quinoline-8-sulfonyl)piperidin-3-amine
3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-2,1-benzoxazole
2-(adamantan-1-yl)-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylacetamide
methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl){[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
5-{2-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
7-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-ethyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}-1H-pyrazole
1-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}-3-methoxypiperidine
ethyl 1-[4-(4H-1,2,4-triazol-4-yl)benzamido]cyclobutane-1-carboxylate
6-ethyl-2-methyl-N-(2-oxoazepan-3-yl)quinoline-4-carboxamide
N4-{[3-(4-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-6-methyl-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
4-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
2-({[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(pyridin-3-ylmethyl)amino)butan-1-ol
2-(2-chloro-4-fluorophenoxymethyl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1,3-oxazole-4-carboxamide
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-(1-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
1-(pyridin-2-ylmethyl)-4-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperazine
5-acetyl-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-2,4-dimethyl-1H-pyrrole-3-carboxamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}cyclooctanamine
2-[(cyclopropylmethyl)sulfanyl]-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)acetamide
methyl({[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl})[1-(pyrazin-2-yl)propan-2-yl]amine
3-[(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)oxy]-N-(2-methoxyethyl)benzamide
4-[(3-methyl-1,2,4-oxadiazol-5-yl)(pyridin-3-yl)methyl]morpholine
1-[(6-methylpyridin-2-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-cyclopentyl-3-(3-methoxyphenyl)-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-2,7,8-trimethylquinoline
2-[4-(dimethylamino)azepane-1-carbonyl]-6-methoxyphenol
3-[5-(5-hydroxypyrazin-2-yl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yloxy)ethyl]acetamide
(1S,3R)-N1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide