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5-(furan-3-ylmethyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
8-(5-ethyl-1,3-oxazole-4-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
3-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
6-chloro-2-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]-1H-1,3-benzodiazole
N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]pent-4-enamide
2-{[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}-6-ethoxyphenol
4-[(2-chloro-4-fluorophenyl)methyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
5-acetyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]thiophene-2-carboxamide
1-(cyclohexylmethyl)-3-methyl-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazole
5-methoxy-2-[2-(2-phenylethyl)morpholine-4-carbonyl]-1,4-dihydropyridin-4-one
6-(propan-2-yloxy)-N4-[2-(pyrrolidin-1-yl)ethyl]pyrimidine-2,4-diamine
4-{4-[2-(propan-2-yloxy)phenyl]-1H-imidazol-2-yl}-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
ethyl 4-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butanoate
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
4-[2-amino-3-cyano-6-(2-methylphenyl)pyridin-4-yl]-N-methylbenzene-1-sulfonamide
N-(isoquinolin-5-ylmethyl)-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[4-(3-{[(2,6-dimethoxypyrimidin-4-yl)amino]methyl}pyridin-2-yl)piperazin-1-yl]ethan-1-one
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(4-ethylphenyl)methyl]piperidin-3-yl}propanamide
(2E)-N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-3-(3-fluorophenyl)-N-(pyridin-3-ylmethyl)prop-2-enamide
{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenol
(3S,4R)-1-(3-methoxy-5-methylthiophene-2-carbonyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
4-(2-fluorophenoxy)-1-(4-methylphthalazin-1-yl)piperidine-4-carboxylic acid
ethyl 4-{2-[4-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}piperidine-1-carboxylate
3-[2-(2-methoxyphenoxy)phenyl]-1-(oxan-4-yl)urea
2-{1-[(3,4-difluorophenyl)methyl]-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
4-({4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzamide
(3R)-1-[7-(5-fluoropyridine-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-ol
2-(2-hydroxyethyl)-6-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
1-[1-(2-cyclohexyl-1,3-benzoxazole-6-carbonyl)piperidin-4-yl]-3-methylbutan-1-ol
1-(3-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}piperidin-1-yl)propan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
6-oxo-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,6-dihydropyridine-3-carboxamide
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]thiophene-2-carboxamide
3-[(dimethylamino)methyl]-1-(5,6-dimethylpyrimidin-4-yl)piperidin-3-ol
methyl 4-{[2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-inden-2-yl]formamido}butanoate
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3-(2-methylpropyl)-1,2-oxazole
4-(2-chloro-6-methoxyphenyl)-N,N-dimethylbenzamide
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(3-fluorophenoxymethyl)piperidine
5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2,4-diol
2-[4-(4-fluorophenyl)-2-[(4-methoxypiperidin-1-yl)methyl]phenoxy]acetic acid
5-(2-fluorophenyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-(1-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-2-phenylethyl)-N-methylpyridine-2-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-ethyl-2-(4-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)acetamide
4-[2-(4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperazin-1-yl)ethyl]morpholine
1-(dimethyl-1,2-oxazole-4-carbonyl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine