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N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
7-(2,2-dimethylpropyl)-2-(1H-indole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-methyl-6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidin-2-amine
5-butyl-4-(3-methoxypyrrolidin-1-yl)-6-methylpyrimidin-2-amine
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-{8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}acetic acid
4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-1-pentylpiperidine
3-(dimethyl-1,2-oxazol-4-yl)-1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}propan-1-one
methyl 2-[1-(5-chloropyridine-2-carbonyl)-3-oxopiperazin-2-yl]acetate
3-(1H-indol-3-ylmethyl)-4-(2-methoxy-5-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)propanamide
1-acetyl-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}piperidine-3-carboxamide
N-(2-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}quinolin-5-yl)acetamide
ethyl(1H-imidazol-2-ylmethyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
(3aR,6aR)-2-cyclopentyl-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
5-methyl-2-(3-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenyl)-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]-2-(propylsulfanyl)ethan-1-one
[5-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)furan-2-yl]methanol
(2-methoxyethyl)[(2-methyl-2H-indazol-3-yl)methyl][(3-methylthiophen-2-yl)methyl]amine
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
4-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-{6-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]pyridin-2-yl}ethan-1-ol
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-3-(2-oxopyrrolidin-1-yl)propanamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperazine
1-(cyclobutylmethyl)-3-hydroxy-3-[(4-methylpiperazin-1-yl)methyl]piperidin-2-one
1-methyl-4-(4-methyl-1H-imidazole-5-carbonyl)-1,4,9-triazaspiro[5.5]undecane
1-[(3-fluorophenyl)methyl]-N-(2-methoxy-2-methylpropyl)-6-oxopiperidine-3-carboxamide
2-(2-aminoethyl)-N-[(2S)-1-methoxypropan-2-yl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
(1S,5R)-6-(2H-1,3-benzodioxole-5-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-2-{4-[4-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
4-(1-ethyl-1H-pyrazole-4-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
[4-({4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}methyl)phenyl]methanol
4-(2-methoxybutanoyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
2-fluoro-5-sulfamoyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)benzamide
7-(2-methoxyethyl)-2-{2-[methyl(phenyl)amino]acetyl}-2,7-diazaspiro[4.5]decan-6-one
N-(1,3-benzoxazol-2-ylmethyl)-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
9-(2-methyl-1H-pyrrole-3-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)[(3-methylpyridin-2-yl)methyl]amine
N-({6-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyridin-3-yl}methyl)acetamide
2-methyl-5-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenol
N-[(2R,3R)-2-hydroxy-1'-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-N,N,6-trimethylpyrimidin-2-amine
2-(ethylamino)-N-{[3-(methylsulfanyl)phenyl]methyl}pyrimidine-5-carboxamide
3-(1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carbonyl)pyridine
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(2-oxoimidazolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
3-{1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
N'-(2,5-dimethylphenyl)-N-[2-(1H-indol-3-yl)ethyl]propanediamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(2-methylpropyl)piperidine-3-carboxamide
methyl 4-({[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amino}methyl)benzoate