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N-[2-(benzylsulfanyl)ethyl]-3-(2-oxoimidazolidin-1-yl)benzamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
2-[(cyclopropylmethyl)sulfanyl]-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}piperidin-3-ol
N-[3-(3-methylphenyl)phenyl]-1-[2-(1H-pyrazol-1-yl)acetyl]piperidine-3-carboxamide
2-[2-(dimethylamino)ethyl]-N-[2-(2-fluorophenyl)ethyl]piperidine-1-carboxamide
methyl({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)[1-(thiophen-2-yl)ethyl]amine
4-{4-[(2,6-difluorophenyl)methyl]piperazin-1-yl}-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[(4-methylphenyl)methyl]-1,4-diazepan-5-one
1-benzyl-5-[(2S)-1-methylpyrrolidin-2-yl]-3-(oxan-4-yl)-1H-1,2,4-triazole
4-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1-[(4-fluorophenyl)methyl]piperazin-2-one
1-(4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-3,5-dimethyl-1H-pyrrol-2-yl)ethan-1-one
7-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-methyl-8-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-{2-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}-N-(2-ethylphenyl)piperidine-1-carboxamide
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-(azocan-1-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}propanamide
N2-(isoquinolin-5-ylmethyl)-N2,N4-dimethylpyrimidine-2,4-diamine
(2-oxo-2-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethyl)urea
(3R)-3-phenyl-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}butan-1-one
1-{3-[2-(4-ethylpiperazin-1-yl)ethyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl}cyclopropane-1-carboxamide
2-({[3-(furan-2-yl)phenyl]methyl}(methyl)amino)-N-methylpropanamide
(1R,3S)-7-(3-fluoro-4-methoxybenzoyl)-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
3-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}-3,4-dihydro-2H-1λ6,2-benzothiazine-1,1-dione
5-{2-[2-(butan-2-yl)phenoxy]acetyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
(2S,4S)-1-(cyclopentylmethyl)-N-ethyl-4-[3-(5-methyl-1H-pyrazol-1-yl)propanamido]pyrrolidine-2-carboxamide
(1R,5R)-N,N-dimethyl-6-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[1-(1H-indol-5-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzene-1-sulfonamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(thiophen-2-yl)butanamide
4-(pyridin-3-yl)-N-[1-(thiophen-2-yl)ethyl]pyrimidin-2-amine
N-[(2-tert-butyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetamide
8-methoxy-2-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1H-pyrazol-1-yl)butan-1-one
{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
2-[1-methyl-4-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
2-[2-(4-phenyl-1H-imidazol-5-yl)-1H-pyrrol-1-yl]pyridine
N-[(3S,4R)-1-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-N-[(3,4,5-trimethoxyphenyl)methyl]-1,3-thiazol-2-amine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
2-methoxy-1-[1'-(piperidin-3-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
(3S)-N,N-dimethyl-1-[4-(trifluoromethyl)pyrimidin-2-yl]azepan-3-amine
7-(3-phenyl-1H-pyrazole-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-methyl-N-(pyrimidin-4-ylmethyl)-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide