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8-[2-(4-ethylpiperazin-1-yl)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-[3-(2,5-dimethoxyphenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
7-[ethoxy(phenyl)methyl]-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-[(4-methyl-1H-imidazol-5-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-{[1-(1-acetylpiperidin-4-yl)pyrrolidin-3-yl]methyl}benzamide
N-methyl-4-phenyl-N-(pyrazin-2-ylmethyl)butanamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]({[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl})methylamine
3-[5-(5-cyanopyridin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-(2-hydroxyethyl)propanamide
1-benzyl-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S)-1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxamide
[1-(3-chloro-5-methoxybenzoyl)-3-ethylpiperidin-3-yl]methanol
1-methyl-3-[2-(piperidin-1-ylmethyl)phenyl]-1-[1-(pyridin-3-yl)propyl]urea
2-[(4aR,7aS)-6,6-dioxo-4-(piperidine-1-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
1-({1-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]cyclopropyl}methyl)-1H-imidazole
1-[(4aS,8aR)-2-oxo-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridine-6-carbonyl]cyclopropane-1-carbonitrile
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[4-(4-fluorophenyl)oxane-4-carbonyl]pyrrolidin-3-yl]methanol
2-amino-4-{4-[1-(dimethylamino)ethyl]phenyl}-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-{1-[2-(1H-pyrrol-1-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)butan-2-ol
N-cyclopentyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
(2S,4S)-4-amino-1-[3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)propanoyl]-N-methylpyrrolidine-2-carboxamide
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-4-acetamido-N-(furan-2-ylmethyl)benzamide
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]ethan-1-one
[(4-ethyl-5-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
2-[4-(2-methyl-5-propylpyrimidin-4-yl)-1H-pyrazol-1-yl]-N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]acetamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
ethyl 1-(5-methoxyfuran-2-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylate
3-(3-methoxyphenoxymethyl)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidine
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-(1,2-oxazol-5-ylmethyl)piperidin-2-one
2-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-6-methylquinolin-4-ol
2-{3-methyl-5-[2-(morpholin-4-yl)phenyl]-1H-1,2,4-triazol-1-yl}acetic acid
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridin-4-one
1-(3-fluorobenzoyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
N-[(2-methylphenyl)methyl]-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
N-(3-methylbutyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
4-ethyl-3-(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]acetamide
2-[4-(2,6-dimethylquinoline-3-carbonyl)piperazin-1-yl]phenol
(1S,5R)-6-benzyl-3-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4S)-4-(dimethylamino)-1-(3-phenylpropyl)pyrrolidin-3-ol
1-benzyl-4-{[4-(pyrrolidine-1-carbonyl)-1,3-oxazol-2-yl]methyl}piperazine
4-[2-(2-chloro-4-fluorophenyl)acetyl]-1-(4-methoxyphenyl)-5-methylpiperazin-2-one
1-methyl-3-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-1-[2-(pyridin-4-yl)ethyl]urea
(2S)-1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-hydroxy-2-phenylethan-1-one
(2R,3R)-1'-[(2-aminopyridin-3-yl)methyl]-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol