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N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
3-(benzenesulfonyl)-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)propanamide
2-(3-chloro-4-hydroxyphenyl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
(2R)-1-({4-[(3-cyanothiophen-2-yl)carbamoyl]phenyl}methyl)pyrrolidine-2-carboxamide
4-{[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]carbamoyl}pyridin-1-ium-1-olate
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(pyrrolidine-1-carbonyl)-decahydro-1,6-naphthyridin-2-one
5,6-dimethoxy-2-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,2-dihydroisoquinolin-1-one
(1S,6R)-9-(ethanesulfonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
4-[2-(piperidine-1-carbonyl)-1-benzofuran-5-yl]-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-ol
2-(benzyloxy)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
8-chloro-2-({methyl[1-(pyridin-3-yl)propyl]amino}methyl)quinolin-4-ol
3-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-1-(2-methylphenyl)urea
4-({2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}methyl)-1-methylpiperidin-4-ol
N-[3-(dimethylamino)phenyl]-3-({[5-(hydroxymethyl)furan-2-yl]methyl}amino)-5-(pyrrolidine-1-sulfonyl)benzamide
1-[(3-methoxyphenyl)methyl]-N-[2-(5-methylfuran-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-ethyl-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-methylpiperidine-3-carboxamide
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazole
(2E)-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-3-(pyridin-3-yl)prop-2-enamide
1-{3-[2-(2,3-dihydro-1-benzofuran-5-yl)pyridin-4-yl]pyrrolidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N-{2-[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]ethyl}acetamide
1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-4-phenoxypiperidine-4-carboxylic acid
N-butyl-6-oxo-N-(3-phenylprop-2-yn-1-yl)-1,6-dihydropyridine-2-carboxamide
(3aR,5R,6S,7aS)-2-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-octahydro-1H-isoindole-5,6-diol
(3S,4R)-1-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
(1R,5S,6R)-6-({[(2-chloropyridin-3-yl)methyl](methyl)amino}methyl)-N,N-diethyl-3-azabicyclo[3.1.0]hexane-3-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]propanamide
4-[(3-fluorophenyl)methyl]-3-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]piperazin-2-one
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(trifluoromethyl)phenyl]urea
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
7-(2-methoxyethyl)-2-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-(1-propyl-1H-pyrazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
2-(4-fluoro-2-methylphenyl)-1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-1H-imidazole
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(quinolin-4-ylmethyl)amine
N-methyl-2-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)butanamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-4-(pyridin-4-yl)pyrimidin-2-amine
N-(2,6-dimethylphenyl)-3-[(2-methylpyrrolidin-1-yl)methyl]benzamide
6-methoxy-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}pyrimidin-4-amine
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-(propoxymethyl)pyrrolidine
6-{2-[(4-ethylpiperidin-1-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
(3S,4R)-3-benzyl-1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-methylpiperidin-4-ol
(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)-N-(2-phenylethyl)pyrrolidine-1-carboxamide
7,7-dimethyl-2-[3-(2-methylpropyl)-1,2-oxazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-methoxy-N-({1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-3-yl}methyl)benzene-1-sulfonamide
(3S,7S)-5-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
methyl 2-{[(3-fluorophenyl)methyl]sulfamoyl}-6-(1-methylcyclopropanecarbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(6-methylpyridin-3-yl)-5-oxopyrrolidine-3-carboxylic acid