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4-({2-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
(1R,9S)-5-amino-3-[3-(pyridin-2-yl)phenyl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
1-(4-hydroxypiperidin-1-yl)-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propan-1-one
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine
3-(2-amino-1,3-thiazol-4-yl)-1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]propan-1-one
(4aS,8aR)-6-(1-ethyl-1H-pyrazole-5-carbonyl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
2-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-N-methylbenzamide
ethyl 3-[(4-fluorophenyl)methyl]-1-[3-(2-methoxyphenyl)propanoyl]piperidine-3-carboxylate
1-(carbamoylmethyl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
3-[ethyl({[3-(3-methoxyphenyl)phenyl]methyl})amino]-1λ6-thiolane-1,1-dione
2-[(methylcarbamoyl)methyl]-3-oxo-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)piperazine-1-carboxamide
1-(3-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-oxopropyl)azepan-2-one
(4aR,7aS)-1-(2-methoxyethyl)-4-[4-(thiophen-2-yl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4R)-4-benzamido-N,N-diethyl-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
2-(furan-2-yl)-5-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)pyrimidine
methyl[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl](oxan-2-ylmethyl)amine
2-(dimethylamino)-2-(3-methylphenyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
6-methyl-2-[3-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N-{4-[({1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}amino)methyl]phenyl}acetamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(4-hydroxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{4-[(dimethylamino)methyl]phenyl}-5-(morpholine-4-sulfonyl)benzoic acid
5-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-3-(4-methoxyphenyl)-1H-pyrazole
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
methyl 5-(2,3-dihydro-1-benzofuran-7-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-[1-(1H-indol-4-ylmethyl)piperidin-4-yl]piperidin-4-ol
1-{1'-[(2-ethylpyrimidin-5-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-[(8-methoxy-2H-chromen-3-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperidin-3-amine
2-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
2-[(4aR,7aS)-4-[(4-chloro-2-fluorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
(3R,5S)-N-[2-(2-ethoxyphenyl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
1-(2-fluorophenyl)-4-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine
N-{[6-(4-methoxy-2-methylphenyl)pyridin-3-yl]methyl}acetamide
2-(3-methoxypropyl)-9-(2-phenoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-{methyl[1-(2-phenylethyl)piperidin-3-yl]carbamoyl}butanoate
8-[(4-ethoxyphenyl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-ethyl-4-{3-[(2-phenylethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
1-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)urea
N-({3-[1-(2-hydroxypropyl)-1,2,3,6-tetrahydropyridin-4-yl]-1,2,4-oxadiazol-5-yl}methyl)-N-methylpyrrolidine-1-carboxamide
N-(2-hydroxybutyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
1-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidine-3-carboxamide
1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
3-{2-[({5-[1-(prop-2-en-1-yl)-1H-pyrazol-3-yl]thiophen-2-yl}methyl)amino]ethyl}-1,3-oxazinan-2-one
1-(cyclohexylmethyl)-N3-ethyl-4-oxo-N5-[phenyl(pyridin-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
[4-({1-[(3-methylquinoxalin-2-yl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
4-(1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)pyridine
2-(cyclopropylmethyl)-9-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-5-propyl-1,3,4-oxadiazole-2-carboxamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-5-propyl-1,2-oxazole-3-carboxamide
5-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}-2-methoxyphenol