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1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
N-(furan-2-ylmethyl)-8-methoxy-N-(pyridin-2-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2-oxoazepan-3-yl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
6-(2-fluorophenyl)-N2-(4-methylphenyl)-1,3,5-triazine-2,4-diamine
(3R,5S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(pyrrolidine-1-carbonyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-(3-chlorobenzoyl)piperidine
2-propyl-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-1,3-thiazole-4-carboxamide
1-cyclopentyl-N-[(1-ethyl-1H-indazol-3-yl)methyl]-5-oxopyrrolidine-3-carboxamide
5-[(isoquinolin-5-yloxy)methyl]-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
5-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]pyridin-2-yl}isoquinoline
4-(oxolane-3-carbonyl)-N,N-diphenylpiperazine-1-carboxamide
(3S,4S)-4-propyl-1-(3-propyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
5-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-1H-indazole
1-[3-(piperidine-1-carbonyl)phenyl]-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
2-{4-[(2,5-dimethylthiophen-3-yl)sulfonyl]morpholin-3-yl}acetic acid
N-(pyridin-3-ylmethyl)-4-(pyrimidin-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-hydroxy-2-(4-methoxyphenyl)-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]acetamide
2-methoxy-6-(2-methyl-1H-imidazol-4-yl)-N,N-bis(propan-2-yl)benzamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-butyl-N-methyl-1,3-benzoxazole-5-carboxamide
3-(3-methyl-1H-1,2,4-triazol-5-yl)-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
2-(4-hydroxyphenyl)-2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}acetic acid
4-methyl-N-[2-(5-methylthiophen-2-yl)ethyl]-1H-imidazole-2-carboxamide
1-acetyl-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)piperidine-4-carboxamide
N-ethyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
[(3-chloro-4-ethoxyphenyl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
4-{1-propyl-5-[3-(1H-pyrazol-4-yl)propyl]-1H-1,2,4-triazol-3-yl}benzamide
3-(cyclopropylmethyl)-1-(2-oxo-1,2-dihydroquinazoline-4-carbonyl)piperidine-3-carboxylic acid
2-(1-butyl-1H-pyrazol-4-yl)-7-fluoro-N,N-dimethylquinoline-4-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(4-chlorophenyl)-4-[2-(pyridin-2-yl)ethyl]morpholine
2-(3-hydroxypropyl)-9-(2-methyl-1,3-thiazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]propan-1-one
(3S,4R)-1-{[3-(morpholin-4-yl)phenyl]methyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
(5S,9aS,9bS)-5-(isoquinolin-5-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-(diethylsulfamoyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperidine-3-carboxamide
2-(3-methoxybenzenesulfonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2-methylpropyl)-1,2-oxazole-3-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-5-phenyl-1,2-oxazole-4-carboxamide
2-cyclopentyl-1-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)ethan-1-one
N-(1-benzylpiperidin-4-yl)-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
N-{1-[1-(2-aminoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
2-(butylsulfanyl)-6-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]pyrimidin-4-amine
N-(4-chloro-2-fluorophenyl)-4-(trifluoroacetyl)-1,4-diazepane-1-carboxamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl][(2,6-difluoro-4-methoxyphenyl)methyl]methylamine
N-{2-[1-(pyridin-2-ylmethyl)-1H-1,2,3-triazol-4-yl]quinolin-6-yl}acetamide
1-ethyl-8-[(4-methoxyphenyl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-methyl-2-oxopentanamide
N-(4-fluoro-2-methylphenyl)-2-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}acetamide
2-({4-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-8-methyl-4H-pyrido[1,2-a]pyrimidin-4-one