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3-(3-chlorophenyl)-N,N-dimethyl-3-phenylpropanamide
3-{4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-1,4,6-trimethyl-1,2-dihydropyridin-2-one
1,3-dimethyl-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-propyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
N-ethyl-6-[3-(methoxymethyl)pyrrolidin-1-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
N-[1-(furan-2-yl)ethyl]-N-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N-methyl-N-(pyrazin-2-ylmethyl)-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(naphthalen-1-ylmethyl)acetamide
3-(6-cyanopyridin-2-yl)benzoic acid
4-[2-(2-chlorophenyl)ethyl]-11-[methyl(1,3-thiazol-4-ylmethyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]acetic acid
N-benzyl{[7-(1H-imidazol-1-yl)-2,3-dihydro-1,4-benzodioxin-6-yl]amino}sulfonamide
8-(5-ethylpyrimidin-2-yl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-(1H-imidazol-1-yl)propyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
N-(2-methoxyethyl)-1,6-dimethyl-N-(pyridin-4-ylmethyl)-1H-indole-2-carboxamide
(1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}piperidin-2-yl)methanol
4-(2-chlorophenoxy)-1-{imidazo[1,2-a]pyridine-3-carbonyl}piperidine
8-(7-methoxy-4-methylquinolin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
(2R)-2-amino-N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}-2-phenylacetamide
3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
1-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-amine
(3S)-1-[4-(dimethylamino)naphthalene-1-carbonyl]-N,N-dimethylazepan-3-amine
1-[3-(4-propylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-(azocan-1-yl)-3-[2-methoxy-5-({[3-(morpholin-4-yl)propyl]amino}methyl)phenoxy]propan-2-ol
3-chloro-4-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)phenol
2-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-1,3-thiazole-4-carboxamide
4-chloro-N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]cyclopropane-1-carboxamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
3-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,6-dimethyl-1,4-dihydroquinolin-4-one
1-(adamantan-2-yl)-4-[(4-fluorophenyl)methyl]-1,4-diazepan-5-one
N,N-diethyl-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
8-fluoro-3-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
N-benzyl-3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carboxamide
4-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-6-(morpholin-4-yl)pyrimidin-2-amine
3-(2,3-dimethylphenyl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[4-(2-chlorophenyl)-3-oxopiperazine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
5-ethyl-N-[1-(6-methylpyridin-2-yl)propan-2-yl]pyrimidin-2-amine
2-amino-1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
1-(4-{[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]methyl}thiophen-2-yl)ethan-1-one
3-(4-cyano-4-phenylpiperidin-1-yl)-N-[(4-methylphenyl)methyl]propanamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyridin-4-ylsulfanyl)acetamide
3-fluoro-N-methyl-N-(1-methylpyrrolidin-3-yl)imidazo[1,2-a]pyridine-2-carboxamide
2-(4-fluorophenyl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-(furan-2-ylmethyl)piperidine
5-chloro-3-[3-(morpholine-4-carbonyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-[(2-chlorophenyl)methyl]-9-(cyclopropylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
8-(1-benzoxepine-4-carbonyl)-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-chloro-N,N-diethyl-3-({methyl[(3-methylpyridin-4-yl)methyl]carbamoyl}amino)benzamide