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1-methyl-3-[4-(morpholine-4-carbonyl)phenyl]-1-(pyridin-3-ylmethyl)urea
5-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl](methyl)[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]amine
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)butanamide
5-[2-(2-phenylethyl)piperidine-1-carbonyl]-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
4-(3-{4-phenyl-5-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}propyl)morpholine
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)ethan-1-one
3-[4-(difluoromethoxy)-2-methylphenyl]-1-[1-(3-methylpyridin-2-yl)propan-2-yl]urea
N,1-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
{4-[(dimethylamino)methyl]-1-{[4-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl}methanol
6-chloro-2-(2-ethoxyethyl)-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
1-[2-(1,4-oxazepan-4-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methoxypyrimidine
(4aS,7aR)-1-[(2-methoxyphenyl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-(cyclohexylmethyl)-4-(cyclopropylmethyl)piperazin-2-yl]ethan-1-ol
1-(5-chlorothiophene-2-carbonyl)-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methyloxolane-2-carboxamide
ethyl 1-[6-(1-benzothiophen-3-yl)-3-{[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]carbamoyl}pyridin-2-yl]piperidine-3-carboxylate
2-[(4aR,7aS)-4-[(2-methylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
(3R,9aR)-8-(3,5-dichlorobenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(5-propyl-1,3,4-oxadiazole-2-carbonyl)piperazin-2-one
N-(propan-2-yl)-2-{[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}acetamide
1-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-2-(2-methyl-1H-indol-3-yl)ethan-1-one
1-{1-[2-(2-ethylphenoxy)ethyl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-2-ylmethyl)piperazine
5-methyl-4-[({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)amino]thieno[2,3-d]pyrimidine-6-carboxylic acid
3-(4-phenoxyphenyl)propanamide
1-methyl-N-[(2-methylphenyl)(pyridin-4-yl)methyl]-1H-pyrazole-4-carboxamide
3-cyclopropyl-N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-5-carboxamide
5-[5-(ethylcarbamoyl)pyridin-2-yl]thiophene-2-carboxylic acid
2-{3-[2-(methylsulfanyl)pyrimidin-4-yl]phenoxy}propanamide
4-[5-(5-ethyl-1,2-oxazole-3-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
{[(3S,4R)-1-(1-benzofuran-2-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
2-[(4-benzylpiperazin-1-yl)methyl]-N,N-bis(prop-2-en-1-yl)-1,3-oxazole-4-carboxamide
1-[(2-methoxyphenyl)methyl]-6-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]piperidine-3-carboxamide
(2R)-N-[2-methyl-4-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-5-oxopyrrolidine-2-carboxamide
2-(5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
2-[4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-(1-benzothiophene-2-carbonyl)-2-(4-methylpiperazine-1-carbonyl)piperazine
[(3R,4R)-1-(2,3-difluoro-4-methoxybenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
3-[1-(2,4-dimethoxybenzoyl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-ethyl-N-(2-methylprop-2-en-1-yl)-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-(azocan-1-yl)-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}ethan-1-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,N-dimethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-sulfonamide
ethyl 1-[(2,5-dimethoxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
5-(1H-indol-1-ylmethyl)-N-[2-(pyridin-3-yloxy)ethyl]-1H-pyrazole-3-carboxamide
3-[(dimethylamino)methyl]-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidin-3-ol