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N-[(6-hydroxypyrimidin-4-yl)methyl]-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
(3aS,6aS)-2-[(2-chloro-4,5-diethoxyphenyl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2,1,3-benzoxadiazole-5-carboxamide
N2-(4-ethyl-5-methylpyrimidin-2-yl)-N1-(pyridin-3-yl)ethane-1,2-diamine
7-(2-methylbenzoyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
5-methyl-5-(4-methylpent-3-en-1-yl)-1-(pyridin-4-ylmethyl)piperidin-2-one
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-2,6-dimethylquinoline
8-(1H-indol-3-ylmethyl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-ethyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}urea
4-[(1S)-1-phenylpropyl]-3-(pyridin-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(pentan-2-yl)-8-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl](quinolin-3-ylmethyl)amine
(1S,5R)-3-(5-chloro-2-methoxybenzenesulfonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
7-fluoro-2-methyl-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)quinoline-4-carboxamide
2-cycloheptyl-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-imidazol-1-yl)-2,3-dihydro-1λ6-thiophene-1,1-dione
N-{[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
2-(3-phenylpropyl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
7-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-{1-[3-(4-hydroxypiperidin-1-yl)propyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
N-benzyl-5-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-ylmethyl]pyrimidin-2-amine
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-methyl-1,4-diazepan-5-one
2-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
3-benzyl-4-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperazin-2-one
3-fluoro-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzene-1-sulfonamide
N-methyl-1-(3-methylbutyl)-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-ethyl-5-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyrimidin-2-amine
1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-(pyridin-3-yl)piperazine
3-{4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-4,5,6-trimethyl-1,2-dihydropyridin-2-one
2-(dimethylamino)-N-(2-methyl-5-{[methyl(oxan-2-ylmethyl)carbamoyl]amino}phenyl)acetamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-3-(furan-2-yl)-3-phenylpropanamide
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-(pyridin-4-ylmethyl)pyridin-2-amine
4-[1-(pyridin-4-ylmethyl)piperidin-4-yl]pyrimidine
1-[1-(4-carbamoyl-1,3-thiazol-2-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
N-ethyl-2-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1,8-naphthyridine-3-carboxamide
5-methyl-3-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydroquinazolin-4-one
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(3-methoxyphenyl)methyl]-N-methylbenzamide
3-{5-[(4-cyclohexyl-1,4-diazepan-1-yl)methyl]thiophen-3-yl}prop-2-yn-1-ol
1-(1H-1,3-benzodiazole-5-carbonyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-{1-[1-(4-chloro-2-fluorobenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-2-ylsulfanyl)acetamide
3-phenyl-N-{1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
6-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-methylpyrimidin-4-ol
3-methyl-7-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
[3-(3-methylbut-2-en-1-yl)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl]methanol
4-methyl-N-{2-methyl-5-[2-(pyrrolidin-1-yl)propanamido]phenyl}benzamide
(3S)-1-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]pyrrolidin-3-ol
2-(2-chlorophenyl)-N,3-dimethyl-N-[(5-methylfuran-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-(2-{3-[3-(6-methoxypyrimidin-4-yl)phenyl]-1H-pyrazol-1-yl}ethyl)morpholine