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N-{4-[1-(quinolin-3-yl)-1H-imidazol-2-yl]phenyl}acetamide
(3S,4R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-{1-[1-(3-acetamidobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(4-methylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-({[(3R,4R)-1-(2-chloro-3-methylbenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
3-{[(benzylsulfamoyl)amino]methyl}-1λ6-thiolane-1,1-dione
4,6-dimethyl-1-(2-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}ethyl)-1,2-dihydropyrimidin-2-one
2-methyl-6-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-3-yl)pyrimidin-4-ol
(2-methoxyethyl)({[2-(methoxymethyl)pyrimidin-5-yl]methyl})[(3-methylthiophen-2-yl)methyl]amine
N-(3-methoxypropyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}propan-1-one
1-[3-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)phenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]propanamide
methyl (2S)-1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
ethyl 4-benzyl-1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxylate
1-[1-(morpholine-4-sulfonyl)-4-phenylpiperidin-4-yl]ethan-1-one
1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-ethyl-1,4-diazepan-5-one
4-[4-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-1H-1,2,3-triazol-1-yl]-1-(2-methoxyethyl)pyrrolidin-2-one
2,2-dimethyl-1-[7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
1-(2-{2-cyclopentyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-[(3S,4S)-4-hydroxy-1-(3-phenylpropyl)pyrrolidin-3-yl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-amino-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1H-1,2,4-triazole-5-carboxamide
N-[(3,4,5-trimethoxyphenyl)methyl]-2,3-dihydro-1H-indene-1-carboxamide
2-methyl-N-(3-{1H-pyrazolo[3,4-b]pyridin-1-yl}phenyl)propanamide
N-(cyclopropylmethyl)-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[1-(4-fluorophenyl)pyrrolidin-3-yl]methyl}-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
3-(1-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)propan-1-ol
(4aS,8aR)-6-(4-chloro-3-fluorobenzoyl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
8-{[3-methoxy-4-(pyrrolidin-1-yl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
1-[(1R,5R)-6-{[3-(benzyloxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-{5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
(2R,3R)-3-amino-1'-[5-(hydroxymethyl)furan-2-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
methyl 9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-3-(naphthalen-2-ylmethyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
3-methanesulfonyl-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
1-[(3,4-dimethylphenyl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
5-fluoro-N-[3-(methylsulfanyl)propyl]quinazolin-4-amine
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-[2-(pyridin-3-yl)ethyl]pyridin-2-amine
ethyl 2-(4-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)acetate
2-[4-(3-ethyl-1H-pyrazole-4-carbonyl)morpholin-3-yl]-N-(4-methoxy-2-methylphenyl)acetamide
(benzylsulfamoyl)[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]amine
methyl 3-{[2-(2H-1,3-benzodioxol-5-yl)acetamido]methyl}-5-(2-fluorobenzamido)benzoate
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}propanamide
2-cyano-N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]benzamide
N-(pyridin-3-ylmethyl)-4-{thieno[2,3-d]pyrimidin-4-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
(4aS,8aR)-6-(1,2-oxazole-5-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[2-(1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
2-{[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
[(2S,4R)-4-(dimethylamino)-1-(quinolin-2-ylmethyl)pyrrolidin-2-yl]methanol