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(1R,3S)-3-amino-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}cyclohexane-1-carboxamide
8-chloro-2-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}quinolin-4-ol
2-[(5-methylpyrazin-2-yl)methyl]-9-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(1-methyl-1H-imidazol-2-yl)-1-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1H-1,2,3-triazole
1-{1-[6-(2,3-difluorophenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-[(4-methoxyphenyl)methyl]pyrimidine
N-(3-phenylpropyl)azepane-4-carboxamide
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[4-(1H-pyrazol-4-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
1-(carbamoylmethyl)-N-[(7-methyl-1H-indol-2-yl)methyl]piperidine-4-carboxamide
methyl 2-{[(2-methoxyphenyl)methyl]amino}pyridine-4-carboxylate
1-{6-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]pyridin-3-yl}ethan-1-one
methyl 3-cyclohexaneamido-6-[(4-phenylpiperazin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
1-cyclohexyl-4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
(1R,5R)-6-(cyclobutylmethyl)-3-(3,4-difluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonane
2-methyl-N-(2-{7-[2-(phenylsulfanyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
3-(2-methylphenyl)-1-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-ol
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperidine
N,1,3-trimethyl-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(naphthalen-1-ylmethyl)pyrrolidin-3-yl]methanol
1-(2-methoxyethyl)-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[1-(2,2-dimethylpropyl)pyrrolidin-2-yl]-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]thiophene-2-carboxamide
2-{[6-(2,3-dihydro-1,4-benzodioxin-6-yl)pyridazin-3-yl]amino}ethan-1-ol
(2S)-2-(3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)-3-phenylpropanamide
(1S,6R)-3-{5-methylthieno[2,3-d]pyrimidin-4-yl}-3,9-diazabicyclo[4.2.1]nonane
(2S,4S)-N-ethyl-4-[3-(methylsulfanyl)propanamido]-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
2-(5-fluoro-2-methoxyphenyl)-2-(4-methyl-3-oxopiperazin-1-yl)acetic acid
3-(2-fluorophenyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
4-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-2-amine
N3-ethyl-N3-(2-methylprop-2-en-1-yl)-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(diethylamino)-2-(furan-2-yl)ethyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
N-[2-(dimethylamino)ethyl]-N-methyl-1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidin-3-amine
4-(5-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
3-[2-(4-methoxyphenyl)ethyl]-N,N-dimethylpiperidine-1-sulfonamide
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(5-methylfuran-2-yl)methyl]piperidine
2-(3,4-dimethoxyphenyl)-3-[(4-ethylpiperazin-1-yl)methyl]-7-methylquinoline
3-(hydroxymethyl)-N-[2-(propylsulfanyl)phenyl]morpholine-4-carboxamide
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(pyrrolidin-1-yl)benzamide
N-[1-(1-cyclopentylpiperidin-4-yl)-1H-pyrazol-5-yl]-4-phenylbutanamide
7-(2-methoxyethyl)-2-(3-methylthiophene-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
6-(hydroxymethyl)-N-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]-1,4-oxazepane-4-carboxamide
4-(oxolane-2-carbonyl)-7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl[3-(5-methylfuran-2-yl)butyl]{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
ethyl 1-(1H-indazole-3-carbonyl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
N-[1-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)propyl]-3-methoxyaniline
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)pyrrolidine-2-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
(3S,7S,8aS)-7-{[(5-chlorothiophen-2-yl)methyl]amino}-3-[(1R)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}pyridine-3-carboxylic acid
1-(4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)-1H-1,2,3,4-tetrazole
N,1,3-trimethyl-N-[3-(piperidin-1-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine