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N-[1-(2-phenylethyl)piperidin-3-yl]-3-(pyridin-2-yl)propanamide
6-ethyl-4-{4-[(methylsulfanyl)methyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(pyridin-4-yl)quinoline-4-carboxamide
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-2-(methylamino)ethan-1-one
2-methyl-5-{[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]sulfanyl}-1,3,4-thiadiazole
1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(3-fluorophenyl)methyl]piperazine
4-(4-{[4-(1H-imidazol-1-yl)phenyl]methyl}morpholine-2-carbonyl)piperazin-2-one
(2-{[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl][(3-methylthiophen-2-yl)methyl]amino}ethyl)dimethylamine
(3aS,6aS)-2-methyl-5-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 1-[2-(4-methoxyphenyl)ethyl]-5-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(furan-2-ylmethyl)-N-[(6-methylquinolin-5-yl)methyl]piperidine-3-carboxamide
1-[(2-aminopyrimidin-5-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N,N-dimethyl-7-(1-methylpiperidine-3-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1,3-dimethyl-5-[2-oxo-2-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)ethyl]imidazolidine-2,4-dione
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[5-(propan-2-yl)-1H-pyrazol-3-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3-carboxamide
ethyl 4-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)piperazine-1-carboxylate
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
4-oxo-4-[3-(2-phenylacetyl)piperidin-1-yl]butane-1-sulfonamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-2-(morpholine-4-carbonyl)pyridin-4-amine
[(2S,4R)-4-(dimethylamino)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}pyrrolidin-2-yl]methanol
ethyl 1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate
2-{[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl][(4-fluorophenyl)methyl]amino}butan-1-ol
3-methyl-8-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{1-cyclohexyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2-methoxyphenol
1-cyclopentanecarbonyl-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]piperidine-4-carboxamide
methyl 2-(1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-3-oxopiperazin-2-yl)acetate
4-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
1-(2-methylpropyl)-5-oxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrrolidine-3-carboxamide
N-[2-(pyrazin-2-yl)ethyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N2,N2,N4,5,6-pentamethylpyrimidine-2,4-diamine
4-{4-[2-(3-methoxypropyl)piperidine-1-carbonyl]-2-methylphenyl}morpholine
2-[1-(2,3-dimethylbenzoyl)pyrrolidin-3-yl]benzoic acid
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(3-methoxypropyl)piperidine
1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-1,2-dihydroquinoxalin-2-one
(1S,6R)-9-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)acetamide
[(2S,4R,5R)-5-(2-fluorophenyl)-4-{[(1H-indol-2-ylmethyl)amino]methyl}-1-methylpyrrolidin-2-yl]methanol
2-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-2-oxo-N-phenylacetamide
4-(1,5-dimethyl-1H-indazole-3-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
4-chloro-3-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1H-pyrazol-5-amine
2-(4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)pyrimidine
1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
5-{4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
7-methyl-2-(thiophen-3-yl)-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1-methyl-1H-imidazol-2-yl)[1-(3-phenylpropyl)piperidin-4-yl]methanol
4-(3-{2-azabicyclo[2.2.1]heptane-2-carbonyl}piperidin-1-yl)-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-[(4-ethyl-1,4-diazepan-1-yl)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N4-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N4,6-dimethyl-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine