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N-[(2-aminopyrimidin-5-yl)methyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methylbenzamide
(1s,4s)-4-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]cyclohexan-1-ol
3-{4-oxo-4-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrol-1-yl]butyl}-3,4-dihydroquinazolin-4-one
5-{[(6-methylhept-5-en-2-yl)amino]methyl}adamantan-2-ol
1-{4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-3-hydroxypropan-1-one
[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl][1-(1H-imidazol-1-yl)propan-2-yl]amine
N-methyl-N-[2-(oxan-2-yl)ethyl]-4-sulfamoylbenzamide
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-(naphthalen-2-yl)piperazine
N-benzyl-N,1-dimethyl-5-{[3-(morpholin-4-yl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-{1-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]piperidin-4-yl}-2-methylpyrimidin-4-ol
{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
4-(4-chlorophenyl)-1-[3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperidin-4-ol
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
[(3R,4R)-1-[(2,5-dichlorophenyl)methyl]-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
3-{1-[(5-fluoro-2-methoxyphenyl)methyl]azetidin-3-yl}pyridine
6-(3,5-dimethoxyphenyl)-N2,N2-diethylpyrimidine-2,4-diamine
1-(adamantan-2-yl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-({4-[(dimethylamino)methyl]phenyl}methyl)-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
1-[(4-fluorophenyl)methyl]-3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]urea
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
3-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]urea
5-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-2,1,3-benzoxadiazole
N-[4-(oxan-2-ylmethoxy)phenyl]morpholine-4-carboxamide
(4aS,8aR)-6-(4,6-dimethylpyrimidin-2-yl)-1-[3-(1H-imidazol-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
N-{[3-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
8-chloro-2-({methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)quinolin-4-ol
(4aR,7aS)-1-{2-[(3-hydroxy-2,2-dimethylpropyl)(methyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
1-(2-methylpropyl)-8-(propan-2-yl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-4-methyl-1-(1-phenylcyclohexanecarbonyl)piperidine-3,4-diol
N-(3-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-oxopropyl)methanesulfonamide
4-(1-acetylpiperidin-4-yl)-6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
4-(2,6-dimethylpyridin-3-yl)-N-(1H-1,2,4-triazol-3-ylmethyl)pyrimidin-2-amine
N-[4-(pyridin-2-yl)butyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
8-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
ethyl 4-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-4-(1,3-thiazol-2-yl)piperazine-1-carboxamide
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[2-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
N-(piperidin-4-ylmethyl)-3-[(1H-pyrazol-3-ylmethyl)sulfamoyl]benzamide
3-{[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-benzothiazole
1-(2-aminoethyl)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]acetamide
N-[3-(4-fluorophenyl)phenyl]-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
4-(2-fluoro-5-methylphenoxy)-1-(quinoxalin-2-yl)piperidine-4-carboxylic acid
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[3-(pyridin-3-yl)propyl]benzamide
8-(cyclopropylmethyl)-N-(4-ethylphenyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
3-methyl-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
{[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]sulfamoyl}dimethylamine