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5,6,7-trimethoxy-3-[(2-methylpyrrolidin-1-yl)methyl]-1,2-dihydroquinolin-2-one
methyl 1-[(4-{[3-(2-hydroxyethoxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperidine-2-carboxylate
N'-cyclopentyl-N-(5-oxo-1-propylpyrrolidin-3-yl)butanediamide
7-[4-hydroxy-4-(hydroxymethyl)azepane-1-carbonyl]quinolin-8-ol
[(dimethyl-1,2-oxazol-4-yl)methyl]({[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl})methylamine
8-(2-ethylbenzoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]-2-(trifluoromethyl)morpholine
(3R,4R)-3,4-dimethyl-1-(5-methyl-2-phenylfuran-3-carbonyl)pyrrolidin-3-ol
ethyl 1-(1H-indol-2-ylmethyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
2,3-dimethyl-6-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
(3R,5S)-1-benzyl-N-(4-fluorophenyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3,4-dihydro-2H-1-benzopyran-6-carboxamide
N2-(pyridin-3-yl)-N1-(thian-4-yl)ethane-1,2-diamine
5-{5-[1-(furan-2-ylmethyl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
2-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}quinolin-4-ol
1,3-dimethyl-2,6-dioxo-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-N,N-dimethylpropane-1-sulfonamide
2-[(4-chlorophenyl)methyl]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,3-benzoxazole-5-carboxamide
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
2-{4-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]morpholin-3-yl}acetic acid
1-{4-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
N-(butan-2-yl)-3-(2-methyl-1H-1,3-benzodiazol-1-yl)-N-(pyridin-4-ylmethyl)propanamide
[(4aS,8aR)-6-(4-ethyl-5-methylpyrimidin-2-yl)-decahydro-1,6-naphthyridin-4a-yl]methanol
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-ethyl-1,2-oxazole-5-carboxamide
1-(4,4-difluoropiperidin-1-yl)-2-(dimethylamino)-2-(3-fluorophenyl)ethan-1-one
methyl N-[4-(4-methoxy-2,5-dimethylphenyl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]carbamate
N-[(1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]acetamide
2-{4-[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}acetamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-6-(propan-2-yl)pyrimidin-4-amine
2-[(dimethylamino)methyl]-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1,3-thiazole-4-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-ethyl-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-indole-5-carboxamide
N-{4-[2-(pyrrolidin-1-yl)acetamido]phenyl}pentanamide
2-({3-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]phenyl}amino)acetic acid
N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
2-(1H-1,3-benzodiazol-2-ylmethoxy)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-hydroxy-N,4-dimethylpentanamide
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[(5-methylfuran-2-yl)methyl]amine
1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-4-(pyrrolidine-1-carbonyl)piperidine
2-{2-[4-(3-chloro-5-fluoro-4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]propyl}pyrazine
2-benzyl-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3-thiazole-4-carboxamide
(3S)-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-amine
3-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methylpyridine-3-carbonitrile
1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]-2-(pyridin-3-yloxy)ethan-1-one
4-methoxy-N-({1-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
methyl 5-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pentanoate
4-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-ethyl-1H-pyrazole
(2R)-2-({3-fluoro-6-methylimidazo[1,2-a]pyridin-2-yl}formamido)propanamide
3-(1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole