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4-(morpholin-4-yl)-6-[4-(oxan-4-yl)piperazin-1-yl]pyrimidin-2-amine
2-[2-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)phenoxy]acetic acid
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(2-methylphenyl)propan-1-one
N-methyl-1-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-(3,5-dimethyl-4-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-1H-pyrrol-2-yl)ethan-1-one
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(piperidine-1-carbonyl)piperidine
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]morpholine-2-carboxamide
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
4-{4-[(2-hydroxyethyl)(methyl)amino]benzoyl}-1-(4-methylphenyl)piperazin-2-one
1-(azocan-1-yl)-3-[2-methoxy-5-({[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-[1-(4-fluorophenyl)propyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-(4-fluoro-3-methylphenyl)urea
1-(2-{[2-amino-6-(propan-2-yl)pyrimidin-4-yl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
4-{imidazo[1,2-a]pyrimidine-2-carbonyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-(1,4-dithiepan-6-yl)-N-(4-fluorophenyl)piperidin-3-amine
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
6-(pyrrolidin-1-ylmethyl)-4-{thieno[3,2-d]pyrimidin-4-yl}-1,4-oxazepan-6-ol
5-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}isoquinoline
8-fluoro-2-{[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]methyl}-1,4-dihydroquinolin-4-one
(4aS,7aR)-1-(3-methoxybenzenesulfonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-ethyl-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(4-cyclopentylphenyl)-2-(thiomorpholin-4-yl)acetic acid
2-{3,5-dimethyl-4-[(4-phenylazepan-1-yl)methyl]-1H-pyrazol-1-yl}ethan-1-ol
2-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-2,7-diazaspiro[4.5]decane
6-[(diethylamino)methyl]-N-(naphthalen-2-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-ethyl-4-[5-(8-hydroxyquinolin-2-yl)-4-phenyl-1H-imidazol-1-yl]pyrrolidin-2-one
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzenesulfonamide
4-methyl-2-[3-(1H-pyrazol-3-yl)phenyl]pyridine
1-(4-fluorophenyl)-4-[(4-methoxy-3-{2-[1-(thiophene-2-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine
1-[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]-3-methoxypropan-1-one
2-benzyl-9-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1-methanesulfonylpiperidin-4-yl)-3-(3-methylphenyl)-1H-pyrazole-4-carboxamide
5-{1-[(4-fluorophenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl}-4-methyl-1,2,3-thiadiazole
(3aS,6aS)-2-{[3-(difluoromethoxy)phenyl]methyl}-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-1-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]urea
1-methyl-3-(3-methylcinnolin-5-yl)-1-[1-(3-methylpyridin-2-yl)propan-2-yl]urea
1-[1-(pent-4-enoyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
5-{4-[(4-cyclohexyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2-methyl-1,4-dihydropyridin-4-one
methyl 2-{1-[5-acetamido-1-ethyl-2-(2-fluorophenyl)-1H-1,3-benzodiazole-7-carbonyl]-3-oxopiperazin-2-yl}acetate
2-{[(2-methylphenyl)methyl]sulfanyl}-N4-[2-(morpholin-4-yl)ethyl]pyrimidine-4,6-diamine
5-[2-(cyclohexylmethyl)morpholine-4-carbonyl]-4-phenylpyrimidin-2-amine
(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-[(3-methoxyphenyl)methyl]piperidin-3-yl)methanol
N-[(2R,4R,6S)-2-cyclohexyl-6-(2,6-dimethylphenyl)oxan-4-yl]acetamide
1-[2-(dimethylamino)ethyl]-4-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}pyrrolidin-2-one
3-{[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-hydroxy-2-methylpropan-1-one
(4aS,7aR)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{2-[1-(3-methylpyridin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
3-{[1-(2-butoxyacetyl)pyrrolidin-3-yl]methyl}benzamide