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4-(2,4-difluorophenyl)-3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-ethyl-5-methylthiophene-3-carbonyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
(1S,5R)-6-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(3S)-3-ethylmorpholin-4-yl]-2-[methyl(piperidin-4-yl)amino]ethan-1-one
2-hydroxy-4-methoxy-N-[(1-methylpyrrolidin-3-yl)methyl]benzamide
2-benzyl-5-formamido-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,1-dimethyl-1H-1,3-benzodiazole-7-carboxamide
6-(3,3-diphenylpiperidine-1-carbonyl)-2,3,4,5-tetrahydropyridazin-3-one
N-(3-hydroxy-3-phenylpropyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[2-(1H-pyrazol-1-yl)benzoyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-(3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)acetic acid
N-(furan-2-ylmethyl)-N-methyl-3-(4-methylpiperazine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
3-{5-benzoyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-[2-(dimethylamino)ethyl]propanamide
(1R,2R,6S,7S)-4-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
6-ethyl-N-methyl-2-oxo-N-[1-(pyridin-3-yl)pentyl]-1,2-dihydropyridine-4-carboxamide
3-{[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
6-{1-[(6-phenoxypyridin-3-yl)methyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
N-methyl-N-(oxan-2-ylmethyl)-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
7-(ethanesulfonyl)-4-(1,4-oxazepan-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
2-(4-methyl-1,4-diazepan-1-yl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}acetamide
4-(1-ethyl-1H-pyrazole-3-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[3-(2-oxopyrrolidin-1-yl)propyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
ethyl 2-(1-{[2-(4-methoxyphenyl)ethyl]carbamoyl}piperidin-2-yl)acetate
(1S,5R)-3-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-(methylamino)pyridine-4-carboxamide
3-(cyclopentylsulfamoyl)-5-(4-hydroxyphenyl)benzoic acid
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(5-ethylfuran-2-yl)methyl]piperidin-3-yl}propanamide
4-[(1-ethyl-5-oxopyrrolidin-3-yl)sulfamoyl]-N-(2-methoxyethyl)benzamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}acetamide
3-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-2-methylphenol
4-{[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]sulfanyl}pyridine
4-(hydroxymethyl)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidin-4-ol
4-{2-[2-(furan-3-yl)-1H-imidazol-1-yl]ethyl}-2-(propan-2-yl)-1,3-thiazole
N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-bromobenzamide
3-(2-oxo-2-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethyl)-1,3-oxazolidin-2-one
N-methyl-3-{[(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)carbamoyl]amino}benzamide
(3S,4S)-1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
1-(4-chlorophenyl)-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)cyclobutane-1-carboxamide
3-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propanoic acid
methyl 2-chloro-4-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)carbamoyl}amino)benzoate
2-{1-[(3,4-difluorophenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-2-(3-methyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)acetamide
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]urea
5-{4-[1-(piperidin-1-yl)ethyl]phenyl}furan-2-carboxamide
8-[(5-methylfuran-2-yl)methyl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3R,4S)-4-cyclopropyl-1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)pyrrolidin-3-amine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide